SCHEMBL4758

SCHEMBL4758

Cc1noc(-c2ccc(Br)cc2)c1/C(=C/CCO)c1ccc(Cc2ccccc2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IP6K1 Q92551 1/20 0.40
IP6K3 Q96PC2 1/20 0.40
IP6K2 Q9UHH9 1/20 0.40
BRD4 O60885 1/20 0.34
L3MBTL1 Q9Y468 3/20 0.34
RAB9A P51151 2/20 0.34
LMNA P02545 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
TRPA1 O75762 1/20 0.34
NPC1 O15118 1/20 0.33
FLT1 P17948 1/20 0.33
MEN1 O00255 1/20 0.32
HTT P42858 1/20 0.32
KMT2A Q03164 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
LPAR1 Q92633 1/20 0.32
GAA P10253 1/20 0.32
NR1H4 Q96RI1 1/20 0.32
SLC6A9 P48067 1/20 0.31
PPARD Q03181 5/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1736 0.92 NR1H4 (0.35) L3MBTL1RAB9ALMNASMN1; SMN2TRPA1
SCHEMBL3368 0.87 IP6K1 (0.39) IP6K1IP6K3IP6K2SMN1; SMN2TRPA1
SCHEMBL7197 0.85 TBXAS1 (0.39) BRD4SMN1; SMN2TRPA1NR1H4TBXAS1
SCHEMBL7735 0.75 MEN1 (0.34) RAB9ANPC1MEN1KMT2A
SCHEMBL1633 0.74 NR1H4 (0.33) SMN1; SMN2TRPA1NPC1NR1H4
SCHEMBL1294 0.69 MEN1 (0.34) SMN1; SMN2NPC1MEN1KMT2A
SCHEMBL1463 0.68 TSHR (0.47) L3MBTL1RAB9ALMNASMN1; SMN2NPC1
SCHEMBL13701 0.67 BRD4 (0.36) IP6K1IP6K3IP6K2BRD4L3MBTL1
SCHEMBL14777651 0.67 BRD4 (0.36) IP6K1IP6K3IP6K2BRD4L3MBTL1
SCHEMBL8250811 0.67 PTPN1 (0.36) RAB9ASMN1; SMN2NPC1MEN1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2483251-A2 POLYCYCLIC COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS Amira Pharmaceuticals, Inc. (US) 2012-08-08 EP disclosed
WO-2011041462-A2 POLYCYCLIC COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS, INC. (US) 2011-04-07 WO disclosed