SCHEMBL3372144

SCHEMBL3372144

CCC(C)[N]Cc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 3/20 0.43
ALDH1A1 P00352 2/20 0.43
CYP3A4 P08684 1/20 0.43
MIF P14174 1/20 0.43
HPGD P15428 1/20 0.43
TP53 P04637 1/20 0.42
TAAR1 Q96RJ0 4/20 0.40
SIGMAR1 Q99720 4/20 0.40
SLC6A2 P23975 2/20 0.40
MAOA P21397 1/20 0.40
SLC6A4 P31645 1/20 0.40
SLC6A3 Q01959 1/20 0.40
CYP2A6 P11509 1/20 0.40
ADORA2A P29274 1/20 0.40
ADORA1 P30542 1/20 0.40
NOS2 P35228 1/20 0.39
SLC18A2 Q05940 1/20 0.38
CYP2D6 P10635 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11876381 0.81 TRPA1 (0.48) TRPA1ALDH1A1CYP3A4MIFHPGD
SCHEMBL1326974 0.79 TAAR1 (0.44) TRPA1ALDH1A1CYP3A4MIFHPGD
SCHEMBL2098954 0.76 NOS2 (0.45) TRPA1ALDH1A1CYP3A4MIFHPGD
SCHEMBL3934527 0.74 MIF (0.45) TRPA1ALDH1A1CYP3A4MIFHPGD
SCHEMBL7871906 0.74 MIF (0.45) TRPA1ALDH1A1CYP3A4MIFHPGD
SCHEMBL8136632 0.74 TAAR1 (0.42) TRPA1ALDH1A1CYP3A4MIFHPGD
SCHEMBL94934 0.68 LMNA (0.38) TRPA1ALDH1A1MIFTP53TAAR1
SCHEMBL8926501 0.68 ESR1 (0.39) TRPA1ALDH1A1CYP3A4MIFHPGD
Ethylbenzene SCHEMBL27526815 0.67 TP53 (0.74) TRPA1TP53TAAR1SIGMAR1SLC6A2
SCHEMBL2145 0.67 ALDH1A1 (0.50) TRPA1ALDH1A1CYP3A4MIFHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4954499-A Pyridazinone derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1990-09-04 US claimed
US-20100324091-A1 Pyrazolone Derivative KOWA COMPANY, LTD. (JP) 2010-12-23 US disclosed
EP-2172458-A1 PYRAZOLONE DERIVATIVE Kowa Company, Ltd. (JP) 2010-04-07 EP disclosed
US-4954499-A Pyridazinone derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1990-09-04 US disclosed
US-4688059-A 3-ARYL(OR HETEROARYL)-3-(OXY OR THIO)PHTHALIDE AS REAGENT IN CARBONLESS DUPLICATING SYSTEM THE HILTON-DAVIS CHEMICAL CO. (US) 1987-08-18 US disclosed
US-4661605-A CARBONLESS CUPLICATION AND THERMAL MARKING SYSTEMS THE HILTON-DAVIS CHEMICAL CO. (US) 1987-04-28 US disclosed
US-4535172-A FOR CARBONLESS DUPLICATING AND THERMAL MARKING SYSTEMS THE HILTON-DAVIS CHEMICAL CO. (US) 1985-08-13 US disclosed
US-4528136-A Process for preparing 2-[bis(aryl)methyl]benzoic acids THE HILTON-DAVIS CHEMICAL CO. (US) 1985-07-09 US disclosed
US-4399291-A CONDENSATION OF A BENZALDEHYDE, AN ANILINE, AN AMINOBENZOIC ACID; OXIDATION STERLING DRUG INC. (US) 1983-08-16 US disclosed
EP-0082394-A2 A process for the production of aminophthalides and amino benzoic acids STERLING DRUG INC. (US) 1983-06-29 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100324091-A1 Pyrazolone Derivative SERPINE1, SERPINC1, TFPI TRPA1 929/4885ALDH1A1 517/4885CYP3A4 710/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.