SCHEMBL7905671

SCHEMBL7905671

Cc1cn2cc(Cc3ccc(N)cc3)cc(-c3cccc(Cl)c3)c2n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 2/20 0.39
DHFR P00374 2/20 0.36
MAOB P27338 3/20 0.36
CCNB2 O95067 1/20 0.36
CCNE2 O96020 1/20 0.36
CDK1 P06493 1/20 0.36
CDK4 P11802 1/20 0.36
CCNB1 P14635 1/20 0.36
CCND1 P24385 1/20 0.36
CCNE1 P24864 1/20 0.36
CDK2 P24941 1/20 0.36
CCNB3 Q8WWL7 1/20 0.36
TLR8 Q9NR97 1/20 0.35
PDE4B Q07343 3/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2C19 P33261 2/20 0.35
TAAR1 Q96RJ0 1/20 0.35
DPP4 P27487 1/20 0.35
DPP8 Q6V1X1 1/20 0.35
DPP9 Q86TI2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3378478 0.87 DHFR (0.39) PDE4DDHFRTLR8DPP4DPP8
SCHEMBL3377783 0.84 PDE4D (0.61) PDE4DPDE4BCYP3A4CYP2C19ADORA1
SCHEMBL3459398 0.83 SMN1; SMN2 (0.35) PDE4DDHFRMAOBCYP3A4CYP2C19
SCHEMBL3380430 0.82 MAOB (0.38) DHFRMAOBCYP2C19DPP4DPP8
SCHEMBL3433258 0.81 DPP4 (0.38) PDE4DDHFRMAOBTLR8PDE4B
SCHEMBL3377436 0.81 HDAC6 (0.39) PDE4DDHFRMAOBCYP3A4TAAR1
SCHEMBL3377711 0.80 KMT2A (0.40) PDE4DPDE4BCYP3A4CYP2C19ADORA1
SCHEMBL3428353 0.79 RAB9A (0.40) PDE4DDHFRMAOBTAAR1TDO2
SCHEMBL3380818 0.78 PDE4D (0.40) PDE4DKDM4EHPGDHTTNPC1
SCHEMBL7915990 0.76 ADORA1 (0.38) TLR8CYP3A4ADORA2AADORA1ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059838-A2 PDE4 INHIBITORS SELECTIVE FOR THE LONG FORM OF PDE4 FOR TREATING INFLAMMATION AND AVOIDING SIDE EFFECTS DECODE GENETICS EHF (IS) 2010-05-27 WO disclosed
WO-2010059836-A1 SUBSTITUTED AZA-BRIDGED BICYCLICS FOR CARDIOVASCULAR AND CNS DISEASE DECODE GENETICS EHF (IS) 2010-05-27 WO disclosed