SCHEMBL3433258

SCHEMBL3433258

Cc1nc2c(-c3cccc(Cl)c3)cc(Cc3ccc(N)cc3)cn2c1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 2/20 0.38
DPP8 Q6V1X1 1/20 0.38
DPP9 Q86TI2 1/20 0.38
PDE4D Q08499 2/20 0.38
DHFR P00374 2/20 0.36
MAOB P27338 2/20 0.35
TLR8 Q9NR97 1/20 0.35
PDE4B Q07343 3/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2C19 P33261 2/20 0.35
TAAR1 Q96RJ0 1/20 0.35
LMNA P02545 2/20 0.34
MAPT P10636 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
RAB9A P51151 1/20 0.34
CYP19A1 P11511 1/20 0.34
TDO2 P48775 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
ABL1 P00519 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3379679 0.88 DHFR (0.38) DPP4DPP8DPP9PDE4DDHFR
SCHEMBL3380528 0.84 PDE4D (0.60) PDE4DPDE4BCYP3A4CYP2C19LMNA
SCHEMBL3379685 0.83 DPP4 (0.39) DPP4DPP8DPP9DHFRMAOB
SCHEMBL7916793 0.83 DPP4 (0.39) DPP4DPP8DPP9PDE4BCYP3A4
SCHEMBL7902720 0.83 DPP4 (0.39) DPP4DPP8DPP9DHFRMAOB
SCHEMBL3428353 0.83 RAB9A (0.40) PDE4DDHFRMAOBTAAR1LMNA
SCHEMBL7905671 0.81 PDE4D (0.39) DPP4DPP8DPP9PDE4DDHFR
SCHEMBL3377436 0.76 HDAC6 (0.39) PDE4DDHFRMAOBCYP3A4TAAR1
SCHEMBL3380717 0.76 PIK3CD (0.38)
SCHEMBL3380282 0.74 CYP3A4 (0.39) MAOBCYP3A4CYP2C19RAB9AADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059838-A2 PDE4 INHIBITORS SELECTIVE FOR THE LONG FORM OF PDE4 FOR TREATING INFLAMMATION AND AVOIDING SIDE EFFECTS DECODE GENETICS EHF (IS) 2010-05-27 WO disclosed
WO-2010059836-A1 SUBSTITUTED AZA-BRIDGED BICYCLICS FOR CARDIOVASCULAR AND CNS DISEASE DECODE GENETICS EHF (IS) 2010-05-27 WO disclosed
WO-2010059836-A1 SUBSTITUTED AZA-BRIDGED BICYCLICS FOR CARDIOVASCULAR AND CNS DISEASE DECODE GENETICS EHF (IS) 2010-05-27 WO disclosed