SCHEMBL3387913

SCHEMBL3387913

CC(=O)Nc1ccc(CCOS(C)(=O)=O)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.49
CA2 P00918 4/20 0.49
POLB P06746 3/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C19 P33261 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
HPGD P15428 1/20 0.49
ALDH1A1 P00352 4/20 0.48
KMT2A Q03164 2/20 0.48
MEN1 O00255 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
AOC3 Q16853 1/20 0.48
CA9 Q16790 2/20 0.46
TSHR P16473 1/20 0.46
CA12 O43570 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
MAPT P10636 2/20 0.46
HTT P42858 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8000580 0.86 SMN1; SMN2 (0.49) POLBHPGDALDH1A1KMT2AMEN1
SCHEMBL7996876 0.85 KMT2A (0.49) CA1CA2ALDH1A1KMT2ACA9
SCHEMBL28396867 0.82 AOC3 (0.54) CA1CA2POLBCYP1A2CYP2D6
SCHEMBL27167710 0.81 CYP17A1 (0.51) CA1CA2MMP1MMP2MMP9
SCHEMBL3258334 0.81 CA2 (0.50) CA1CA2ALDH1A1CA9TSHR
SCHEMBL9585898 0.80 ALDH1A1 (0.63) CA1CA2CYP1A2TDP1ALDH1A1
SCHEMBL29622963 0.79 AOC3 (0.67) CA1CA2POLBCYP1A2CYP2C19
SCHEMBL29622962 0.79 AOC3 (0.67) CA1CA2POLBCYP1A2CYP2C19
SCHEMBL11039771 0.79 KMT2A (0.50) CA1CA2HPGDALDH1A1KMT2A
SCHEMBL28890376 0.79 CA2 (0.41) CA1CA2ALDH1A1CA9TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010043633-A1 2H-PYRAZOLO [4,3-D]PYRIMIDIN-5-AMINE DERIVATIVES AS H4 HISTAMINE RECEPTOR ANTAGONISTS FOR THE TREATMENT OF ALLERGIC, IMMUNOLOGICAL AND INFLAMMATORY DISEASES PALAU PHARMA, S. A. (ES) 2010-04-22 WO disclosed