SCHEMBL3393341

SCHEMBL3393341

CN(c1cc(-c2ccc(C#N)cc2Cl)ccn1)c1cc(-c2ccccn2)[nH]n1

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.43
TGFBR1 P36897 4/20 0.42
GRM5 P41594 6/20 0.37
METAP2 P50579 1/20 0.35
METAP1 P53582 1/20 0.35
EGLN2 Q96KS0 2/20 0.34
CRHR1 P34998 1/20 0.33
ACVR1B P36896 1/20 0.33
FFAR1 O14842 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3392062 0.90 KCNH2 (0.54) KCNH2TGFBR1GRM5METAP2METAP1
SCHEMBL3393142 0.84 CYP19A1 (0.41) KCNH2
SCHEMBL3397575 0.81 KCNH2 (0.43) KCNH2TGFBR1EGLN2
SCHEMBL3395600 0.81 L3MBTL1 (0.35) KCNH2TGFBR1GRM5METAP2METAP1
SCHEMBL3397038 0.80 KCNH2 (0.42) KCNH2TGFBR1GRM5EGLN2
SCHEMBL3393337 0.77 KCNH2 (0.58) KCNH2TGFBR1GRM5CRHR1
SCHEMBL3397167 0.77 KCNH2 (0.42) KCNH2EGLN2
SCHEMBL3399143 0.76 KCNH2 (0.41) KCNH2EGLN2
SCHEMBL3392275 0.76 KCNH2 (0.46) KCNH2TGFBR1GRM5METAP2METAP1
SCHEMBL3434735 0.76 KCNH2 (0.40) KCNH2TGFBR1EGLN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010046780-A2 ANTI VIRAL COMPOUNDS INSTITUT PASTEUR KOREA (KR) 2010-04-29 WO disclosed