SCHEMBL3409949

SCHEMBL3409949

COc1cc(Nc2nc(C)cc(-c3ccccc3)n2)ccc1-c1nc(C)c[nH]1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 12/20 0.51
ABCB1 P08183 1/20 0.43
ABCC1 P33527 1/20 0.43
ABCG2 Q9UNQ0 1/20 0.43
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
DOT1L Q8TEK3 1/20 0.41
AGTR1 P30556 1/20 0.41
KCNH2 Q12809 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3410260 0.88 NPC1 (0.53) IMPDH2ABCG2NPC1RAB9ADOT1L
SCHEMBL3411066 0.87 NPC1 (0.47) IMPDH2NPC1RAB9ADOT1LKCNH2
SCHEMBL3406068 0.84 NPC1 (0.46) IMPDH2ABCG2NPC1RAB9ADOT1L
SCHEMBL3408093 0.83 PSEN1 (0.44) IMPDH2ABCB1ABCC1ABCG2NPC1
SCHEMBL3407955 0.83 NPC1 (0.51) IMPDH2ABCG2NPC1RAB9ADOT1L
SCHEMBL3406191 0.82 IMPDH2 (0.45) IMPDH2
SCHEMBL3410316 0.81 IMPDH2 (0.44) IMPDH2ABCG2NPC1RAB9ADOT1L
SCHEMBL3406232 0.80 NPC1 (0.41) IMPDH2NPC1RAB9ADOT1LKCNH2
SCHEMBL3408862 0.80 NPC1 (0.43) IMPDH2ABCG2NPC1RAB9ADOT1L
SCHEMBL3407100 0.80 MAPT (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2257541-A1 MODULATORS FOR AMYLOID BETA F. Hoffmann-La Roche AG (CH) 2010-12-08 EP disclosed
WO-2009103652-A1 MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2009-08-27 WO disclosed