SCHEMBL3408568

SCHEMBL3408568

COc1cc(Nc2nc(C)cc(OC3CCCC3)n2)ccc1-c1nc(C)c[nH]1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
EHMT2 Q96KQ7 10/20 0.39
EHMT1 Q9H9B1 9/20 0.39
KCNH2 Q12809 1/20 0.38
DOT1L Q8TEK3 1/20 0.36
TTK P33981 2/20 0.36
CLK1 P49759 1/20 0.35
CLK2 P49760 1/20 0.35
CAMKK2 Q96RR4 1/20 0.35
PDGFRB P09619 1/20 0.35
PDGFRA P16234 1/20 0.35
IMPDH2 P12268 1/20 0.35
PSEN1 P49768 1/20 0.34
PSEN2 P49810 1/20 0.34
APH1B Q8WW43 1/20 0.34
NCSTN Q92542 1/20 0.34
APH1A Q96BI3 1/20 0.34
PSENEN Q9NZ42 1/20 0.34
PDE7A Q13946 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3412405 0.90 NPC1 (0.39) NPC1RAB9AEHMT2EHMT1KCNH2
SCHEMBL3406068 0.87 NPC1 (0.46) NPC1RAB9AEHMT2EHMT1KCNH2
SCHEMBL3410260 0.84 NPC1 (0.53) NPC1RAB9AEHMT2EHMT1KCNH2
SCHEMBL3410316 0.82 IMPDH2 (0.44) NPC1RAB9AEHMT2EHMT1KCNH2
SCHEMBL3411085 0.82 NPC1 (0.42) NPC1RAB9AEHMT2EHMT1KCNH2
SCHEMBL3410702 0.82 USP2 (0.45) NPC1RAB9AEHMT2EHMT1KCNH2
SCHEMBL3406681 0.80 NPC1 (0.41) NPC1RAB9AEHMT2EHMT1KCNH2
SCHEMBL3407955 0.79 NPC1 (0.51) NPC1RAB9AEHMT2EHMT1KCNH2
SCHEMBL3411061 0.79 SLC2A1 (0.48) NPC1RAB9AEHMT2EHMT1
SCHEMBL3406468 0.79 KCNH2 (0.42) NPC1RAB9AEHMT2EHMT1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2257541-A1 MODULATORS FOR AMYLOID BETA F. Hoffmann-La Roche AG (CH) 2010-12-08 EP disclosed
WO-2009103652-A1 MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2009-08-27 WO disclosed