SCHEMBL3424293

SCHEMBL3424293

O=C(O)[C@]1(C2CCCCC2)CCCN1

nearest known ligand 0.33

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ARG1 P05089 1/20 0.33
ARG2 P78540 1/20 0.33
LMNA P02545 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10659624 1.00 ARG1 (0.33) ARG1ARG2LMNATSHR
SCHEMBL4634034 1.00 ARG1 (0.33) ARG1ARG2LMNATSHR
SCHEMBL10989977 1.00 ARG1 (0.33) ARG1ARG2LMNATSHR
Hydrochloric Acid SCHEMBL3418562 0.98 ARG1 (0.32) ARG1ARG2
SCHEMBL29113103 0.94 LMNA (0.33) LMNATSHR
SCHEMBL11100097 0.94 LMNA (0.33) LMNATSHR
SCHEMBL15664981 0.92 ARG1 (0.34) ARG1ARG2
Hydrochloric Acid SCHEMBL25348469 0.90 ARG1 (0.33) ARG1ARG2
Hydrochloric Acid SCHEMBL25348463 0.90 ARG1 (0.33) ARG1ARG2
SCHEMBL5791673 0.89 LMNA (0.33) LMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 73 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118271224-A Preparation method of (2S, 4S) -4-cyclohexyl-L-proline 浙江华海药业股份有限公司 2024-07-02 CN claimed
CN-110885358-A Vaccine for preventing tumor recurrence and metastasis and application method thereof 浙江爱睦世医学科技有限公司 2020-03-17 CN claimed
CN-108727242-A A kind of preparation method of the trans- -4- cyclohexyl-L-PROLINE of blood-pressure drug key intermediate 常州制药厂有限公司 2018-11-02 CN claimed
CN-104744511-A Fosinopril production method ZHANG YUN 2015-07-01 CN claimed
US-20120142939-A1 PROCESS FOR THE PREPARATION OF FOSINOPRIL AND INTERMEDIATES THEREOF DIPHARMA FRANCIS S.R.L. (IT) 2012-06-07 US claimed
EP-2460808-A1 Process for the preparation of fosinopril and intermediates thereof Dipharma Francis S.r.l. (IT) 2012-06-06 EP claimed
EP-2264039-A1 Process for the preparation of fosinopril and intermediates thereof Dipharma Francis S.r.l. (IT) 2010-12-22 EP claimed
US-20100297711-A1 PROCESS FOR THE SYNTHESIS OF FOSINOPRIL AND INTERMEDIATES THEREOF DIPHARMA FRANCIS S.R.L. (IT) 2010-11-25 US claimed
US-7078532-B2 Process for manufacture of fosinopril sodium LUPIN LABORATORIES LIMITED (IN) 2006-07-18 US claimed
US-20040225127-A1 Process for manufacture of fosinopril sodium LUPIN LABORATORIES LIMITED (IN) 2004-11-11 US claimed
EP-1383779-A2 A PROCESS FOR MANUFACTURE OF FOSINOPRIL SODIUM LUPIN LABORATORIES LIMITED (IN) 2004-01-28 EP claimed
WO-2002088149-A2 A PROCESS FOR MANUFACTURE OF FOSINOPRIL SODIUM LUPIN LABORATORIES LIMITED (IN) 2002-11-07 WO claimed
EP-0437799-B1 The diastereoselective preparation of phosphinate esters SQUIBB & SONS INC (US) 1995-02-22 EP claimed
EP-0437799-A1 The diastereoselective preparation of phosphinate esters E.R. SQUIBB & SONS, INC. (US) 1991-07-24 EP claimed
US-5008399-A Reacting phosphinic acid ester with halo ester in presence of specific base in organic solvent, hydrogenating E. R. SQUIBB & SONS, INC. (US) 1991-04-16 US claimed
EP-4746915-A1 TRIM21-BINDING MOLECULES United Kingdom Research and Innovation (GB) 2026-05-27 EP disclosed
WO-2025021697-A1 TRIM21-BINDING MOLECULES UNITED KINGDOM RESEARCH AND INNOVATION (GB) 2025-01-30 WO disclosed
EP-0053902-A1 Phosphinylalkanoyl substituted prolines E.R. Squibb & Sons, Inc. (US) 1982-06-16 EP disclosed
EP-0052991-A1 Carboxyalkyl amino acid derivatives of various substituted prolines E.R. Squibb & Sons, Inc. (US) 1982-06-02 EP disclosed
US-4316905-A HYPOTENSIVE AGENTS E. R. SQUIBB & SONS, INC. (US) 1982-02-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120142939-A1 PROCESS FOR THE PREPARATION OF FOSINOPRIL AND INTERMEDIATES THEREOF FOS, FOSB, NPPA ARG1 1297/4885ARG2 2480/4885LMNA 1693/4885
US-20040225127-A1 Process for manufacture of fosinopril sodium FOS, FOSB, AGT ARG1 1881/4885ARG2 2931/4885LMNA 2759/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.