SCHEMBL3445191

SCHEMBL3445191

Cc1ncc2c(C)csc2n1

nearest known ligand 0.32

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 3/20 0.32
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
PKM P14618 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
MAPK1 P28482 1/20 0.31
HSD17B10 Q99714 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
HCRTR1 O43613 1/20 0.30
HCRTR2 O43614 1/20 0.30
PDK4 Q16654 2/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1900202 0.80 CYP2A6 (0.32)
SCHEMBL1820304 0.80 CYP2A6 (0.35) ALDH1A1SMN1; SMN2
SCHEMBL6362575 0.72 LMNA (0.46) ALDH1A1MAPTSMN1; SMN2MAPK1L3MBTL1
SCHEMBL30362436 0.71 MRGPRX1 (0.33) ALDH1A1SMN1; SMN2
SCHEMBL8274148 0.71 MRGPRX1 (0.33) ALDH1A1SMN1; SMN2
SCHEMBL7926335 0.68 ALDH1A1 (0.40) ALDH1A1MAPTSMN1; SMN2HSD17B10KMT2A
SCHEMBL19699901 0.68 CYP2A6 (0.34) ALDH1A1SMN1; SMN2KMT2A
SCHEMBL3891533 0.68 RPS6KB2 (0.36) ALDH1A1MAPTSMN1; SMN2L3MBTL1
SCHEMBL17813446 0.67 PDK2 (0.32) PDK2PDK4
SCHEMBL7923181 0.67 KDM4E (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021129737-A1 COMPOUND HAVING KHK INHIBITORY EFFECT 南京明德新药研发有限公司 2021-07-01 WO disclosed
US-20110195957-A1 SUBSTITUTED DIAZEPAN OREXIN RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2011-08-11 US disclosed
US-7816351-B2 5,6-dimethylthieno[2,3-di] pyrimidine derivatives, the preparation method thereof and the pharmaceutical composition comprising the same for anti-virus EQUISPHARM CO., LTD (KR) 2010-10-19 US disclosed
US-20080234482-A1 5,6-Dimethylthieno[2,3-Di] Pyrimidine Derivatives, the Preparation Method Thereof and the Pharmaceutical Composition Comprising the Same for Anti-Virus EQUISPHARM CO., LTD (KR) 2008-09-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080234482-A1 5,6-Dimethylthieno[2,3-Di] Pyrimidine Derivatives, the Preparation Method Thereof and the Pharmaceutical Composition Comprising the Same for Anti-Virus DUS2, DPYD, DUT PDK2 268/4885ALDH1A1 368/4885MAPT 2681/4885
US-20110195957-A1 SUBSTITUTED DIAZEPAN OREXIN RECEPTOR ANTAGONISTS HCRTR2, HCRTR1, CRHR1 PDK2 2210/4885ALDH1A1 3194/4885MAPT 712/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.