SCHEMBL3452132

SCHEMBL3452132

C#CCOc1ccc(CCl)cc1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA12 O43570 6/20 0.50
CA9 Q16790 6/20 0.50
CA4 P22748 5/20 0.50
CA2 P00918 2/20 0.50
CA1 P00915 2/20 0.50
GSTP1 P09211 1/20 0.50
CA7 P43166 1/20 0.50
MAOA P21397 7/20 0.46
MAOB P27338 7/20 0.46
ACHE P22303 1/20 0.46
CYP19A1 P11511 1/20 0.43
PTGS2 P35354 2/20 0.41
HDAC3 O15379 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
NCOR2 Q9Y618 1/20 0.37
POLB P06746 1/20 0.37
MAPK1 P28482 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9503476 0.94 CA12 (0.46) CA12CA9CA4CA2CA1
SCHEMBL5704167 0.84 CA12 (0.63) CA12CA9CA4CA2CA1
SCHEMBL31725844 0.83 CA12 (0.53) CA12CA9CA4CA2CA1
Hydrochloric Acid SCHEMBL21694040 0.82 CA12 (0.61) CA12CA9CA4CA2CA1
SCHEMBL9156553 0.81 CA12 (0.52) CA12CA9CA4CA2CA1
SCHEMBL634485 0.79 FFAR1 (0.38) MAOBCYP19A1HSD17B10
SCHEMBL7381752 0.79 CA12 (0.50) CA12CA9CA4CA2CA1
SCHEMBL3677826 0.79 GSTP1 (0.55) CA12CA9CA4CA2CA1
SCHEMBL19616328 0.79 CA12 (0.50) CA12CA9CA4CA2CA1
SCHEMBL11957426 0.79 CA12 (0.55) CA12CA9CA4CA2CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10953369-B2 Spirocentric compounds and polymers thereof GEORGIA TECH RESEARCH CORPORATION (US) 2021-03-23 US disclosed
US-10926226-B2 Functionalized membranes and methods of production thereof ExxonMobil Research & Engineering Company Company (US) 2021-02-23 US disclosed
EP-3762391-A1 SPIROCENTRIC COMPOUNDS AND POLYMERS THEREOF ExxonMobil Research and Engineering Company (US) 2021-01-13 EP disclosed
WO-2019173646-A1 SPIROCENTRIC COMPOUNDS AND POLYMERS THEREOF EXXONMOBIL RESEARCH AND ENGINEERING COMPANY (US) 2019-09-12 WO disclosed
US-20190275469-A1 Functionalized Membranes and Methods of Production Thereof GEORGIA TECH RESEARCH CORPORATION 2019-09-12 US disclosed
US-20190276454-A1 Spirocentric Compounds and Polymers Thereof GEORGIA TECH RESEARCH CORPORATION 2019-09-12 US disclosed
US-7820818-B2 Heteroaryl nitrile derivatives NOVARTIS AG (CH) 2010-10-26 US disclosed
US-20090227596-A1 HETEROARYL NITRILE DERIVATIVES NOVARTIS AG (CH) 2009-09-10 US disclosed
US-7544688-B2 Hetereoaryl nitrile derivatives NOVARTIS AG (CH) 2009-06-09 US disclosed
EP-1537111-B1 HETEREOARYL NITRILE DERIVATIVES NOVARTIS AG (CH) 2007-05-02 EP disclosed
US-20060142575-A1 Hetereoaryl nitrile derivatives NOVARTIS AG (CH) 2006-06-29 US disclosed
EP-1537111-A1 HETEREOARYL NITRILE DERIVATIVES Novartis AG (CH) 2005-06-08 EP disclosed
WO-2004020441-A1 HETEREOARYL NITRILE DERIVATIVES NOVARTIS AG (CH) 2004-03-11 WO disclosed
EP-0748159-A4 INSECTICIDAL N-(SUBSTITUTED ARYLMETHYL)-4- BIS(SUBSTITUTED PHENYL)METHYL]PIPERIDINES FMC CORP (US) 1997-11-19 EP disclosed
US-5639763-A FOR AGRICULTURAL APPLICATIONS FMC CORPORATION (US) 1997-06-17 US disclosed
EP-0748159-A1 INSECTICIDAL N-(SUBSTITUTED ARYLMETHYL)-4- BIS(SUBSTITUTED PHENYL)METHYL]PIPERIDINES FMC CORPORATION (US) 1996-12-18 EP disclosed
US-5569664-A AGRICULTURAL INSECTICIDES FMC CORPORATION (US) 1996-10-29 US disclosed
WO-1995023507-A1 INSECTICIDAL N-(SUBSTITUTED ARYLMETHYL)-4-[BIS(SUBSTITUTED PHENYL)METHYL]PIPERIDINES FMC CORPORATION (US) 1995-09-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190276454-A1 Spirocentric Compounds and Polymers Thereof PKD1, PKD2, VIM CA12 1262/4885CA9 1424/4885CA4 1744/4885
US-10926226-B2 Functionalized membranes and methods of production thereof LNPK, PLA2G2A, EPCAM CA12 476/4885CA9 1737/4885CA4 1346/4885
US-10953369-B2 Spirocentric compounds and polymers thereof PKD1, PKD2, VIM CA12 1262/4885CA9 1424/4885CA4 1744/4885
US-20090227596-A1 HETEROARYL NITRILE DERIVATIVES CTSK, CTSS, CTSZ CA12 3291/4885CA9 870/4885CA4 509/4885
US-20060142575-A1 Hetereoaryl nitrile derivatives CTSK, CTSZ, CTSE CA12 2378/4885CA9 814/4885CA4 481/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.