SCHEMBL3463370

SCHEMBL3463370

C=CCOC(=O)NNCc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 8/20 0.52
ALDH1A1 P00352 3/20 0.48
CYP3A4 P08684 1/20 0.47
MAPT P10636 1/20 0.45
TSHR P16473 1/20 0.42
HSD17B10 Q99714 1/20 0.42
TGM2 P21980 1/20 0.42
PKM P14618 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
CSNK2A2 P19784 1/20 0.40
CSNK2A1 P68400 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7624194 0.84 CASP1 (0.68) CASP1ALDH1A1CYP3A4MAPT
SCHEMBL7396978 0.82 CA12 (0.57) ALDH1A1SMN1; SMN2KMT2A
SCHEMBL7434407 0.79 GAA (0.60) ALDH1A1MAPTTSHRHSD17B10SMN1; SMN2
SCHEMBL4557754 0.78 GAA (0.63) CASP1ALDH1A1CYP3A4TSHRHSD17B10
SCHEMBL7647656 0.76 TGM2 (0.52) ALDH1A1TGM2SMN1; SMN2KMT2A
SCHEMBL11002529 0.75 CASP1 (0.49) CASP1ALDH1A1CYP3A4MAPTTSHR
SCHEMBL28300827 0.75 SMN1; SMN2 (0.48) CASP1ALDH1A1CYP3A4TSHRHSD17B10
SCHEMBL17895893 0.74 ALDH1A1 (0.56) ALDH1A1CYP3A4TSHRHSD17B10TGM2
SCHEMBL473103 0.74 TDP1 (0.55) ALDH1A1CYP3A4TSHRSMN1; SMN2
SCHEMBL14560262 0.74 CASP1 (0.54) CASP1ALDH1A1CYP3A4MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010010435-A2 FUSED OXAZOLE AND THIAZOLE DERIVATIVES AS TRPMS MODULATORS GLENMARK PHARMACEUTICAL S.A. (CH) 2010-01-28 WO disclosed