SCHEMBL3475862

SCHEMBL3475862

CC(C)(C)OC(=O)N(c1cscn1)S(=O)(=O)c1cc(Cl)c(Oc2ccc(Cl)cc2C2CCN(C(=O)O)C(C(C)(C)C)C2)cc1F

nearest known ligand 0.45

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 19/20 0.45
SCN8A Q9UQD0 1/20 0.39
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
SCN5A Q14524 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1094461 0.87 SCN9A (0.50) SCN9ASCN8ACYP3A4CYP2C9SCN5A
SCHEMBL28074465 0.77 SCN9A (0.41) SCN9ASCN8ACYP3A4CYP2C9SCN5A
SCHEMBL28519988 0.77 SCN8A (0.41) SCN8A
SCHEMBL16094574 0.74 SCN9A (0.41) SCN9ASCN8ACYP3A4CYP2C9SCN5A
SCHEMBL3477862 0.74 SCN9A (0.43) SCN9A
SCHEMBL1743618 0.74 SCN9A (0.49) SCN9ACYP3A4CYP2C9
SCHEMBL17509683 0.74 SCN9A (0.40) SCN9ASCN8ACYP3A4CYP2C9SCN5A
SCHEMBL17523542 0.74 SCN9A (0.39) SCN9ASCN8ACYP3A4CYP2C9SCN5A
SCHEMBL17961886 0.73 SCN9A (0.40) SCN9ASCN8ACYP3A4CYP2C9SCN5A
SCHEMBL18013128 0.73 SCN9A (0.64) SCN9ASCN8ACYP2C9SCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100197655-A1 SULFONAMIDE DERIVATIVES Pfizer Limited Icagen, Inc. 2010-08-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100197655-A1 SULFONAMIDE DERIVATIVES SULT2A1, SULT1A1, TPST2 SCN9A 73/4885SCN8A 32/4885CYP3A4 133/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.