SCHEMBL3477271

SCHEMBL3477271

O=S(=O)(Nc1cscn1)c1cccnc1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SLC40A1 Q9NP59 5/20 0.50
GLO1 Q04760 1/20 0.50
CKS1B P61024 3/20 0.49
SKP2 Q13309 3/20 0.49
KEAP1 Q14145 1/20 0.46
NFE2L2 Q16236 1/20 0.46
KMT2A Q03164 1/20 0.45
CA2 P00918 1/20 0.44
MAPT P10636 1/20 0.44
SCN1A P35498 3/20 0.44
SCN5A Q14524 3/20 0.44
SCN8A Q9UQD0 3/20 0.44
SCN9A Q15858 2/20 0.44
BRD4 O60885 1/20 0.44
NAPRT Q6XQN6 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1093964 0.83 SCN1A (0.54) KEAP1KMT2ASCN1ASCN5ASCN8A
SCHEMBL6292016 0.78 SLC40A1 (0.55) SLC40A1GLO1CKS1BSKP2KEAP1
Formic Acid SCHEMBL19616986 0.77 SCN1A (0.49) KEAP1SCN1ASCN5ASCN8ASCN9A
SCHEMBL22634311 0.75 KMT2A (0.54) SLC40A1KMT2AMAPTSCN1ASCN5A
SCHEMBL30845613 0.75 SCN1A (0.49) SCN1ASCN5ASCN8ASCN9A
SCHEMBL16720161 0.75 SCN1A (0.48) CA2SCN1ASCN5ASCN8ASCN9A
SCHEMBL31017724 0.75 SCN1A (0.44) SCN1ASCN5ASCN8ASCN9A
SCHEMBL11704625 0.74 SMN1; SMN2 (0.56) KMT2AMAPTSCN1ASCN5ASCN8A
SCHEMBL25382203 0.73 SMN1; SMN2 (0.52) SLC40A1GLO1CKS1BSKP2KEAP1
SCHEMBL31017719 0.73 MAPT (0.46) MAPTSCN1ASCN5ASCN8ASCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112638898-B Heteroaryl substituted sulfonamide compounds and their use as sodium channel inhibitors 泽农医药公司 2024-04-09 CN disclosed
US-8907101-B2 Sulfonamide derivatives PFIZER LIMITED (GB) 2014-12-09 US disclosed
US-20130338111-A1 Sulfonamide Derivatives ICAGEN, INC. (US) 2013-12-19 US disclosed
US-20120149679-A1 Sulfonamide Derivatives ICAGEN, INC. 2012-06-14 US disclosed
US-20100197655-A1 SULFONAMIDE DERIVATIVES Pfizer Limited Icagen, Inc. 2010-08-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100197655-A1 SULFONAMIDE DERIVATIVES SULT2A1, SULT1A1, TPST2 SLC40A1 3958/4885GLO1 2222/4885CKS1B 2074/4885
US-20130338111-A1 Sulfonamide Derivatives SULT2A1, SULT1A1, TPST2 SLC40A1 3958/4885GLO1 2222/4885CKS1B 2074/4885
US-20120149679-A1 Sulfonamide Derivatives SULT2A1, SULT1A1, TPST2 SLC40A1 3958/4885GLO1 2222/4885CKS1B 2074/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.