SCHEMBL3482959

SCHEMBL3482959

Cc1ccccc1N1CCN(C(CCOC(N)=O)c2ccc(F)cc2)CC1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 1/20 0.43
P2RX7 Q99572 2/20 0.42
MC4R P32245 1/20 0.41
ADRB2 P07550 1/20 0.41
ADRB1 P08588 1/20 0.41
ADRB3 P13945 1/20 0.41
ADRA1D P25100 1/20 0.41
ADRA1A P35348 1/20 0.41
ADRA1B P35368 1/20 0.41
ABCB1 P08183 3/20 0.40
AVPR1A P37288 1/20 0.39
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39
THRB P10828 1/20 0.39
CCR3 P51677 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3482923 0.89 TP53 (0.50) ADRB2ADRB1ADRB3ADRA1DADRA1A
SCHEMBL3483116 0.87 MEN1 (0.50) MAPT
SCHEMBL3483021 0.83 MC4R (0.46) MC4RTP53MAPTCCR3
SCHEMBL3482581 0.80 ME2 (0.46) MC4RTP53MAPTCCR3
SCHEMBL3482665 0.80 LMNA (0.50) MC4RADRB2ADRB1ADRB3ADRA1D
SCHEMBL3482900 0.79 KMT2A (0.52) MC4RADRB1TP53MAPTCCR3
SCHEMBL3482318 0.79 CYP2C9 (0.42) ADRB2ADRB1ADRB3ADRA1DADRA1A
SCHEMBL2116792 0.76 ADRB1 (0.56) ADRB1
SCHEMBL3482997 0.76 POLB (0.54) MC4RTP53MAPT
SCHEMBL15962306 0.70 SLC6A4 (0.57)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2150550-A1 NOVEL CARBAMOYLOXY ARYL ALKAN ARYLPIPERAZINE COMPOUND, PHARMACEUTICAL COMPOSITIONS COMPRISING THE COMPOUND AND METHOD FOR TREATING PAIN, ANXIETY AND DEPRESSION BY ADMINISTERING THE COMPOUND SK Holdings Co., Ltd. (KR) 2010-02-10 EP disclosed
WO-2008140197-A1 NOVEL CARBAMOYLOXY ARYL ALKAN ARYLPIPERAZINE COMPOUND, PHARMACEUTICAL COMPOSITIONS COMPRISING THE COMPOUND AND METHOD FOR TREATING PAIN, ANXIETY AND DEPRESSION BY ADMINISTERING THE COMPOUND SK HOLDINGS CO., LTD. (KR) 2008-11-20 WO disclosed