SCHEMBL3482318

SCHEMBL3482318

COc1ccc(Cl)cc1N1CCN(C(CCOC(N)=O)c2ccc(F)cc2)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
HTR3E A5X5Y0 1/20 0.42
HTR3B O95264 1/20 0.42
HTR3A P46098 1/20 0.42
HTR3D Q70Z44 1/20 0.42
HTR3C Q8WXA8 1/20 0.42
FFAR4 Q5NUL3 1/20 0.41
ADRA1D P25100 2/20 0.41
ADRA1A P35348 2/20 0.41
ADRA1B P35368 2/20 0.41
MAPT P10636 2/20 0.40
KDM4E B2RXH2 1/20 0.40
MAPK1 P28482 1/20 0.40
LMNA P02545 1/20 0.40
POLB P06746 1/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
SLC6A3 Q01959 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3482923 0.88 TP53 (0.50) ADRA1DADRA1AADRA1BMAPTMAPK1
SCHEMBL3482665 0.87 LMNA (0.50) ADRA1DADRA1AADRA1BMAPTMAPK1
SCHEMBL3483021 0.79 MC4R (0.46) MAPTLMNAPOLBSLC6A2SLC6A4
SCHEMBL3482959 0.79 AOC3 (0.43) ADRA1DADRA1AADRA1BMAPTTP53
SCHEMBL3482900 0.79 KMT2A (0.52) MAPTLMNAPOLBTP53ADRB1
SCHEMBL2116476 0.79 ADRB1 (0.51) ADRA1DADRA1AADRA1BADRB1
SCHEMBL3483116 0.78 MEN1 (0.50) MAPTPOLBSLC6A2SLC6A4
SCHEMBL3482937 0.77 KMT2A (0.50) MAPTMAPK1LMNATP53ADRB1
SCHEMBL3482581 0.75 ME2 (0.46) MAPTKDM4ELMNATP53
SCHEMBL3483019 0.72 MAPT (0.53) MAPTMAPK1LMNATHRBADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2150550-A1 NOVEL CARBAMOYLOXY ARYL ALKAN ARYLPIPERAZINE COMPOUND, PHARMACEUTICAL COMPOSITIONS COMPRISING THE COMPOUND AND METHOD FOR TREATING PAIN, ANXIETY AND DEPRESSION BY ADMINISTERING THE COMPOUND SK Holdings Co., Ltd. (KR) 2010-02-10 EP disclosed
WO-2008140197-A1 NOVEL CARBAMOYLOXY ARYL ALKAN ARYLPIPERAZINE COMPOUND, PHARMACEUTICAL COMPOSITIONS COMPRISING THE COMPOUND AND METHOD FOR TREATING PAIN, ANXIETY AND DEPRESSION BY ADMINISTERING THE COMPOUND SK HOLDINGS CO., LTD. (KR) 2008-11-20 WO disclosed