SCHEMBL3483791

SCHEMBL3483791

O=C(O)NCCCNCCCNC(=O)O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA3 P07451 3/20 0.50
CA5A P35218 3/20 0.50
CA5B Q9Y2D0 3/20 0.50
CA12 O43570 2/20 0.50
CA2 P00918 2/20 0.50
CA4 P22748 2/20 0.50
CA6 P23280 2/20 0.50
CA7 P43166 2/20 0.50
CA9 Q16790 2/20 0.50
CA14 Q9ULX7 2/20 0.50
PAOX Q6QHF9 1/20 0.44
KDM4E B2RXH2 5/20 0.40
KDM1A O60341 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
MAPK1 P28482 1/20 0.38
HIF1A Q16665 1/20 0.38
PRMT1 Q99873 1/20 0.37
CYP2C19 P33261 3/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18338812 0.97 CA3 (0.54) CA3CA5ACA5BCA12CA2
SCHEMBL23069642 0.94 CA12 (0.50) CA3CA5ACA5BCA12CA2
SCHEMBL8958360 0.91 KDM4E (0.43) CA3CA5ACA5BCA12CA2
SCHEMBL20536196 0.90 CA3 (0.43) CA3CA5ACA5BCA12CA2
SCHEMBL20536003 0.90 CA2 (0.43) CA3CA5ACA5BCA12CA2
SCHEMBL4555815 0.88 PAOX (0.63) CA3CA5ACA5BCA12CA2
SCHEMBL13842143 0.88 CA12 (0.52) CA3CA5ACA5BCA12CA2
SCHEMBL16246838 0.88 CA12 (0.52) CA3CA5ACA5BCA12CA2
SCHEMBL18874871 0.86 CA3 (0.45) CA3CA5ACA5BCA12CA2
SCHEMBL719437 0.86 CA12 (0.54) CA3CA5ACA5BCA12CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024091894-A1 PNU ANTHRACYCLINE DERIVATIVES AND METHODS OF USE THEREOF MERCK SHARP & DOHME LLC (US) 2024-05-02 WO disclosed
EP-3271423-B1 CATIONIC DIRECT DYES BASF SE (DE) 2022-08-31 EP disclosed
US-20210087337-A1 COMPOUNDS, COMPOSITIONS AND METHODS RELATED TO ANTIMICROBIAL APPLICATIONS VYOME THERAPEUTICS LIMITED (IN) 2021-03-25 US disclosed
EP-3507325-A2 COMPOUNDS, COMPOSITONS AND METHODS RELATED TO ANTIMICROBIAL APPLICATIONS Vyome Therapeutics Limited (IN) 2019-07-10 EP disclosed
WO-2018042367-A2 COMPOUNDS, COMPOSITONS AND METHODS RELATED TO ANTIMICROBIAL APPLICATIONS VYOME BIOSCIENCES PVT. LTD. (IN) 2018-03-08 WO disclosed
US-8440643-B2 Inhibitors of beta-lactamase METHYLGENE INC. (CA) 2013-05-14 US disclosed
US-20100279983-A1 NOVEL INHIBITORS OF BETA-LACTAMASE METHYLGENE INC. 2010-11-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100279983-A1 NOVEL INHIBITORS OF BETA-LACTAMASE MGAM, MGAM2, PGLS CA3 3852/4885CA5A 3237/4885CA5B 2940/4885
US-20210087337-A1 COMPOUNDS, COMPOSITIONS AND METHODS RELATED TO ANTIMICROBIAL APPLICATIONS CUTA, GMPS, MMP8 CA3 4877/4885CA5A 4679/4885CA5B 4436/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.