SCHEMBL3497780

SCHEMBL3497780

O=C(N[C@@H](Cc1ccccc1)C(=O)O)c1ccc(O)cc1

nearest known ligand 0.72

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 2/20 0.72
CA2 P00918 5/20 0.69
CA1 P00915 5/20 0.69
ACE P12821 2/20 0.64
MME P08473 1/20 0.60
GPR132 Q9UNW8 2/20 0.60
CTSL P07711 1/20 0.60
MEN1 O00255 1/20 0.60
ALDH1A1 P00352 1/20 0.60
KMT2A Q03164 1/20 0.60
CA12 O43570 2/20 0.59
CA9 Q16790 2/20 0.59
HPGDS O60760 1/20 0.59
L3MBTL1 Q9Y468 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8520566 1.00 PTPN1 (0.72) PTPN1CA2CA1ACEMME
SCHEMBL3404637 0.94 CA2 (0.69) PTPN1CA2CA1ACEMME
SCHEMBL8667639 0.94 CA2 (0.69) PTPN1CA2CA1ACEMME
SCHEMBL5793343 0.94 CA2 (0.69) PTPN1CA2CA1ACEMME
SCHEMBL8671997 0.94 CA2 (0.77) PTPN1CA2CA1ACEMME
SCHEMBL4054764 0.94 CA2 (0.77) PTPN1CA2CA1ACEMME
SCHEMBL4054766 0.94 CA2 (0.77) PTPN1CA2CA1ACEMME
SCHEMBL4364597 0.93 PTPN1 (0.64) PTPN1CA2CA1ACEMME
SCHEMBL6513134 0.93 CA2 (0.68) PTPN1CA2CA1ACEMME
SCHEMBL528464 0.90 ACE (0.76) PTPN1CA2CA1ACEMME

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112837763-A Structure search method, structure search device, and recording medium 富士通株式会社 2021-05-25 CN disclosed
CN-111816257-A Combination structure search device, combination structure search method, and medium 富士通株式会社 2020-10-23 CN disclosed
US-20100160241-A1 NOVEL COMPOUND HAVING GPR54 AGONISTIC ACTIVITY KYOTO UNIVERSITY (JP) 2010-06-24 US disclosed
US-5986136-A Photolabeling reagent PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 1999-11-16 US disclosed
EP-0178911-B1 COMPOSITION CONTAINING A PENEM OR CARBAPENEM ANTIBIOTIC SANKYO COMPANY LIMITED (JP) 1992-01-22 EP disclosed
US-4757066-A Reduces renal toxicity SANKYO COMPANY LIMITED (JP) 1988-07-12 US disclosed
EP-0178911-A2 Composition containing a penem or carbapenem antibiotic SANKYO COMPANY LIMITED (JP) 1986-04-23 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100160241-A1 NOVEL COMPOUND HAVING GPR54 AGONISTIC ACTIVITY GPR52, GPR84, GPR4 PTPN1 3022/4885CA2 2475/4885CA1 4606/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.