Doxribtimine

Doxribtimine

SCHEMBL3514796

Cc1cn([C@H]2C[C@H](O)[C@@H](CO)O2)c(=O)[nH]c1=O.O=c1[nH]cnc2nc[nH]c12.[N-]=[N+]=CC(=O)OC[C@H](N)C(=O)O

nearest known ligand 0.48

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

P

The experimentally established mechanism targets of Doxribtimine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.48
TSHR P16473 2/20 0.48
ALB P02768 1/20 0.48
TK1 P04183 1/20 0.48
PKM P14618 1/20 0.48
BLM P54132 1/20 0.48
PMP22 Q01453 1/20 0.48
CYP2D6 P10635 1/20 0.48
ABCG2 Q9UNQ0 3/20 0.43
ABCB1 P08183 1/20 0.43
RNASE1 P07998 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Doxribtimine SCHEMBL9176732 0.92 LMNA (0.52) LMNATSHRALBTK1PKM
Doxribtimine SCHEMBL341619 0.83 LMNA (0.59) LMNATSHRALBTK1PKM
Doxribtimine SCHEMBL2164592 0.82 TK1 (0.53) LMNATSHRALBTK1PKM
Doxribtimine SCHEMBL17985772 0.79 LMNA (0.54) LMNATSHRALBTK1PKM
Doxribtimine SCHEMBL9465657 0.78 TK1 (0.51) LMNATSHRALBTK1PKM
Azaserine SCHEMBL20520234 0.77 ALDH1A1 (0.41) TSHR
Doxribtimine SCHEMBL3166229 0.76 TK1 (0.52) LMNATSHRALBTK1PKM
Doxribtimine SCHEMBL1164058 0.76 TK1 (0.53) LMNATSHRALBTK1PKM
Doxribtimine SCHEMBL8366525 0.76 TK1 (0.53) LMNATSHRALBTK1PKM
Doxribtimine SCHEMBL3155784 0.76 TK1 (0.52) LMNATSHRALBTK1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100279401-A1 T Cell Hybridomas And Related Compositions And Methods For Assaying And Modulating T Cell Receptor-Mediated Immune Responses NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2010-11-04 US disclosed
EP-1802741-A4 T CELL HYBRIDOMAS AND RELATED COMPOSITIONS AND METHODS FOR ASSAYING AND MODULATING T CELL RECEPTOR-MEDIATED IMMUNE RESPONSE UNIV OREGON HEALTH & SCIENCE (US) 2008-03-05 EP disclosed
EP-1802741-A2 T CELL HYBRIDOMAS AND RELATED COMPOSITIONS AND METHODS FOR ASSAYING AND MODULATING T CELL RECEPTOR-MEDIATED IMMUNE RESPONSE Oregon Health and Science University (US) 2007-07-04 EP disclosed
WO-2006010020-A2 T CELL HYBRIDOMAS OREGON HEALTH AND SCIENCE UNIVERSITY (US) 2006-01-26 WO disclosed
EP-0651819-A1 METHODS FOR HUMAN MONOCLONAL ANTIBODY PRODUCTION IMMUNET (US) 1995-05-10 EP disclosed
WO-1993019197-A1 HUMAN MONOCLONAL ANTIBODIES AND METHODS FOR HUMAN MONOCLONAL ANTIBODY PRODUCTION IMMUNET (US) 1993-09-30 WO disclosed
US-4950598-A Process for making T cell hybridomas THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 1990-08-21 US disclosed