SCHEMBL3522362

SCHEMBL3522362

Fc1ccc(-c2nc3cnccn3c2-c2ccncc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIA1 P42261 2/20 0.58
PRKD3 O94806 5/20 0.58
MAPK9 P45984 5/20 0.58
CSNK1A1 P48729 5/20 0.58
CSNK1D P48730 5/20 0.58
PRKD2 Q9BZL6 5/20 0.58
MAP4K4 O95819 4/20 0.58
CSNK1G2 P78368 4/20 0.58
MINK1 Q8N4C8 4/20 0.58
MAP3K20 Q9NYL2 4/20 0.58
CSNK1G3 Q9Y6M4 4/20 0.58
GSK3B P49841 4/20 0.58
FRK P42685 3/20 0.58
MAPK8 P45983 3/20 0.58
FGFR1 P11362 2/20 0.58
CSNK1G1 Q9HCP0 2/20 0.58
PRKCD Q05655 1/20 0.58
ERBB4 Q15303 1/20 0.58
MAPK14 Q16539 7/20 0.56
MAPK13 O15264 4/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12781591 0.96 GRIA1 (0.62) GRIA1PRKD3MAPK9CSNK1A1CSNK1D
SCHEMBL7218478 0.83 PTGS2 (0.60) GRIA1PRKD3MAPK9CSNK1A1CSNK1D
SCHEMBL7221055 0.83 GRIA1 (0.54) GRIA1PRKD3MAPK9CSNK1A1CSNK1D
SCHEMBL9298472 0.83 CSNK1D (0.58) PRKD3MAPK9CSNK1A1CSNK1DPRKD2
SCHEMBL2068605 0.79 TUBB4A (0.53) GRIA1PRKD3MAPK9CSNK1A1CSNK1D
SCHEMBL3521737 0.79 TUBB4A (0.53) GRIA1PRKD3MAPK9CSNK1A1CSNK1D
SCHEMBL3522644 0.78 PRKD3 (0.62) GRIA1PRKD3MAPK9CSNK1A1CSNK1D
SCHEMBL3522717 0.78 CSNK1E (0.66) PRKD3MAPK9CSNK1A1CSNK1DPRKD2
SCHEMBL3525119 0.77 CSNK1D (0.52) GRIA1PRKD3MAPK9CSNK1A1CSNK1D
SCHEMBL108805 0.77 GRIA1 (0.45) GRIA1PRKD3MAPK9CSNK1A1CSNK1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230192699-A1 COMPOUNDS AS CASEIN KINASE INHIBITORS Gritscience Biopharmaceuticals Co., Ltd. (CN) 2023-06-22 US disclosed
US-20230192699-A1 COMPOUNDS AS CASEIN KINASE INHIBITORS Gritscience Biopharmaceuticals Co., Ltd. (CN) 2023-06-22 US disclosed
US-20230192699-A1 COMPOUNDS AS CASEIN KINASE INHIBITORS Gritscience Biopharmaceuticals Co., Ltd. (CN) 2023-06-22 US disclosed
EP-4126878-A1 COMPOUNDS AS CASEIN KINASE INHIBITORS Gritscience Biopharmaceuticals Co., Ltd. (CN) 2023-02-08 EP disclosed
CN-115335057-A Method for inhibiting casein kinase 北京原基华毅生物科技有限公司 2022-11-11 CN disclosed
CN-115298183-A Compounds as casein kinase inhibitors 北京原基华毅生物科技有限公司 2022-11-04 CN disclosed
US-7709468-B2 Imidazo based heterocycles ABBOTT LABORATORIES (US) 2010-05-04 US disclosed
US-7709468-B2 Imidazo based heterocycles ABBOTT LABORATORIES (US) 2010-05-04 US disclosed
US-7709468-B2 Imidazo based heterocycles ABBOTT LABORATORIES (US) 2010-05-04 US disclosed
US-20070099925-A1 Novel imidazo based heterocycles ABBVIE INC. 2007-05-03 US disclosed
US-20070099925-A1 Novel imidazo based heterocycles ABBVIE INC. 2007-05-03 US disclosed
US-20070099925-A1 Novel imidazo based heterocycles ABBVIE INC. 2007-05-03 US disclosed
WO-2007028051-A2 NOVEL IMIDAZO BASED HETEROCYCLES ABBOTT LABORATORIES (US) 2007-03-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070099925-A1 Novel imidazo based heterocycles CDK4, CDK2, MAP3K19 GRIA1 1729/4885PRKD3 365/4885MAPK9 189/4885
US-20230192699-A1 COMPOUNDS AS CASEIN KINASE INHIBITORS CSNK2A3, CSNK1A1, CSNK1G3 GRIA1 2785/4885PRKD3 173/4885MAPK9 62/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.