SCHEMBL3524342

SCHEMBL3524342

COC(=O)CCC#Cc1cc(Cl)ccc1NS(=O)(=O)c1ccc(C)c2ccccc12

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC16A3 O15427 2/20 0.42
SLC16A7 O60669 1/20 0.42
SLC16A8 O95907 1/20 0.42
HTR5A P47898 1/20 0.42
FABP4 P15090 5/20 0.42
ACLY P53396 1/20 0.40
BRD4 O60885 1/20 0.39
CCR9 P51686 1/20 0.38
SLC22A12 Q96S37 1/20 0.38
POLB P06746 1/20 0.37
MAPT P10636 2/20 0.37
NPC1 O15118 1/20 0.37
TSHR P16473 1/20 0.37
MEN1 O00255 1/20 0.36
LMNA P02545 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3519735 0.88 SLC16A3 (0.45) SLC16A3SLC16A7SLC16A8HTR5AACLY
SCHEMBL3524537 0.85 ACLY (0.47) SLC16A3SLC16A7SLC16A8HTR5AACLY
SCHEMBL3522442 0.85 EDNRA (0.42) SLC16A3SLC16A7SLC16A8HTR5AACLY
SCHEMBL3523698 0.83 ERBB2 (0.50) ACLYCCR9MAPTMEN1LMNA
SCHEMBL3523363 0.83 SLC16A3 (0.43) SLC16A3SLC16A7SLC16A8HTR5AACLY
SCHEMBL3526026 0.82 PTGES2 (0.50) ACLYSLC22A12
SCHEMBL3530147 0.82 CYTH2 (0.43) FABP4ACLYCCR9POLBMAPT
SCHEMBL3524790 0.81 SLC22A12 (0.61) ACLYSLC22A12MEN1KMT2A
SCHEMBL3525803 0.81 ALDH1A1 (0.48) CCR9MAPTMEN1LMNAKMT2A
SCHEMBL3527669 0.81 LMNA (0.48) CCR9MAPTLMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8436040-B2 Method of treating conditions involving PPAR-receptors with indole compounds LABORATOIRES FOURNIER S.A. (FR) 2013-05-07 US disclosed
US-20100286137-A1 Method of Treating Conditions Involving PPAR-Receptors with Indole Compounds LABORATORIES FOURNIER S.A. (FR) 2010-11-11 US disclosed
US-7795297-B2 Indole compounds, method of preparing them and uses thereof LABORATORIES FOURNIER S.A. (FR) 2010-09-14 US disclosed
US-20080153816-A1 Indole Compounds, Method of Preparing Them and Uses Thereof LABORATOIRES FOURNIER S.A. (FR) 2008-06-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080153816-A1 Indole Compounds, Method of Preparing Them and Uses Thereof LIPG, GPR119, IAPP SLC16A3 3744/4885SLC16A7 3821/4885SLC16A8 3938/4885
US-20100286137-A1 Method of Treating Conditions Involving PPAR-Receptors with Indole Compounds GPR119, PPARA, PPARG SLC16A3 3322/4885SLC16A7 3308/4885SLC16A8 3304/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.