SCHEMBL3524488

SCHEMBL3524488

O=c1cc(O)c2ccc(Br)cc2o1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 1/20 0.74
ALDH1A1 P00352 4/20 0.68
KDM4E B2RXH2 3/20 0.68
KMT2A Q03164 2/20 0.68
CA12 O43570 2/20 0.59
CA9 Q16790 2/20 0.59
CA1 P00915 1/20 0.59
MEN1 O00255 1/20 0.54
MAPT P10636 1/20 0.54
MET P08581 1/20 0.49
MAOB P27338 2/20 0.48
MCL1 Q07820 4/20 0.46
AKR1B1 P15121 3/20 0.46
HSD17B3 P37058 3/20 0.46
HPGD P15428 2/20 0.46
HSD17B10 Q99714 2/20 0.46
LMNA P02545 1/20 0.46
CYP1A2 P05177 1/20 0.46
GLA P06280 1/20 0.46
GAA P10253 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31290723 1.00 PIM1 (0.74) PIM1ALDH1A1KDM4EKMT2ACA12
SCHEMBL2761544 0.85 PIM1 (1.00) PIM1ALDH1A1KDM4EKMT2ACA12
SCHEMBL23640512 0.82 PIM1 (0.64) PIM1ALDH1A1KDM4EKMT2ACA12
SCHEMBL958685 0.81 ALDH1A1 (1.00) ALDH1A1KDM4EKMT2ACA12CA9
SCHEMBL29419327 0.81 ALDH1A1 (1.00) ALDH1A1KDM4EKMT2ACA12CA9
Water SCHEMBL11848480 0.79 ALDH1A1 (0.96) ALDH1A1KDM4EKMT2ACA12CA9
SCHEMBL8119361 0.78 ALDH1A1 (0.68) PIM1ALDH1A1KDM4EKMT2ACA12
SCHEMBL2761833 0.78 ALDH1A1 (0.68) PIM1ALDH1A1KDM4EKMT2ACA12
SCHEMBL14492920 0.78 ALDH1A1 (0.68) PIM1ALDH1A1KDM4EKMT2ACA12
SCHEMBL5346628 0.78 ALDH1A1 (0.68) PIM1ALDH1A1KDM4EKMT2ACA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 55 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116178385-B Coumarin hemicyanine dye with structural rigidity, and preparation method and application thereof 山西大学 2025-01-28 CN claimed
CN-116178385-A Coumarin hemicyanine dye with structural rigidity, and preparation method and application thereof 山西大学 2023-05-30 CN claimed
CN-106008475-A Coumarin NEDD8 activating enzyme inhibitor 南京工业大学 2016-10-12 CN claimed
EP-4735452-A2 HETEROBIFUNCTIONAL COMPOUNDS FOR THE DEGRADATION OF KRAS PROTEIN Merck Patent GmbH (DE) 2026-05-06 EP disclosed
EP-4735438-A2 HETEROBIFUNCTIONAL COMPOUNDS FOR THE DEGRADATION OF KRAS Merck Patent GmbH (DE) 2026-05-06 EP disclosed
US-20250326732-A1 CHROMEN-2-ONE MODULATORS OF POLRMT PRETZEL THERAPEUTICS, INC. (US) 2025-10-23 US disclosed
CN-116178385-B Coumarin hemicyanine dye with structural rigidity, and preparation method and application thereof 山西大学 2025-01-28 CN disclosed
WO-2025006753-A2 HETEROBIFUNCTIONAL COMPOUNDS FOR THE DEGRADATION OF KRAS PROTEIN MERCK PATENT GMBH (DE) 2025-01-02 WO disclosed
WO-2025006783-A2 HETEROBIFUNCTIONAL COMPOUNDS FOR THE DEGRADATION OF KRAS MERCK PATENT GMBH (DE) 2025-01-02 WO disclosed
CN-115160300-B Coumarin compound, preparation method thereof and application of coumarin compound in resisting Alzheimer disease 中国人民解放军北部战区总医院 2024-05-31 CN disclosed
CN-116178385-A Coumarin hemicyanine dye with structural rigidity, and preparation method and application thereof 山西大学 2023-05-30 CN disclosed
US-20070149579-A1 Novel pharmaceutical compounds MERCK CANADA INC. (CA) 2007-06-28 US disclosed
EP-1531812-B1 FUSED HETEROARYL DERIVATIVES FOR USE AS P38 KINASE INHIBITORS IN THE TREATMENT OF I.A. RHEUMATOID ARTHRITIS SMITHKLINE BEECHAM CORP (US) 2007-06-27 EP disclosed
US-20070054942-A1 Fused heteroaryl derivatives and their use as p38 kinase inhibitors GLAXOSMITHKLINE LLC 2007-03-08 US disclosed
US-20060122221-A1 Fused heteroaryl derivatives for use as p38 kinase inhibitors in the treatment of i.a. rheumatoid arthristis SMITHKLINE BEECHAM CORPORATION 2006-06-08 US disclosed
EP-1531812-A1 FUSED HETEROARYL DERIVATIVES FOR USE AS P38 KINASE INHIBITORS IN THE TREATMENT OF I.A. RHEUMATOID ARTHRISTIS SMITHKLINE BEECHAM CORPORATION (US) 2005-05-25 EP disclosed
WO-2004010995-A1 FUSED HETEROARYL DERIVATIVES FOR USE AS P38 KINASE INHIBITORS IN THE TREATMENT OF I.A. RHEUMATOID ARTHRISTIS SMITHKLINE BEECHAM CORPORATION (US) 2004-02-05 WO disclosed
US-6114546-A Aminomethylene derivatives and ultraviolet absorbent comprising thereof CHEMIPRO KASEI KAISHA, LIMITED (JP) 2000-09-05 US disclosed
EP-0950655-A1 AMINOMETHYLENE DERIVATIVES AND ULTRAVIOLET ABSORBER COMPRISING THE SAME CHEMIPRO KASEI KAISHA, LIMITED (JP) 1999-10-20 EP disclosed
US-3974289-A Coumarin derivatives for the treatment of allergies BEECHAM GROUP LIMITED (EN) 1976-08-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250326732-A1 CHROMEN-2-ONE MODULATORS OF POLRMT POLRMT, TFAM, POLM PIM1 2621/4885ALDH1A1 3178/4885KDM4E 2158/4885
US-20060122221-A1 Fused heteroaryl derivatives for use as p38 kinase inhibitors in the treatment of i.a. rheumatoid arthristis MAPK7, CNKSR1, MAPK1 PIM1 2055/4885ALDH1A1 1269/4885KDM4E 4559/4885
US-20070149579-A1 Novel pharmaceutical compounds LTA4H, LTB4R2, LTC4S PIM1 2670/4885ALDH1A1 431/4885KDM4E 3391/4885
US-20070054942-A1 Fused heteroaryl derivatives and their use as p38 kinase inhibitors MAPK1, MAPK7, MAPKAPK2 PIM1 1126/4885ALDH1A1 2057/4885KDM4E 4697/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.