SCHEMBL3528023

SCHEMBL3528023

N#Cc1ccc(N)cc1-c1ccc(Cl)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.51
MEN1 O00255 5/20 0.51
KMT2A Q03164 5/20 0.51
HPGD P15428 4/20 0.51
MAPT P10636 2/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C19 P33261 1/20 0.51
ALDH1A1 P00352 7/20 0.45
RXFP1 Q9HBX9 2/20 0.45
PPARG P37231 1/20 0.45
STAT3 P40763 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
NR2E3 Q9Y5X4 1/20 0.45
NCOR2 Q9Y618 1/20 0.45
LMNA P02545 2/20 0.44
POLB P06746 1/20 0.44
ADORA2A P29274 3/20 0.43
ADORA1 P30542 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2959360 0.82 CYP11B1 (0.44) KDM4EMEN1KMT2AHPGDMAPT
SCHEMBL2958151 0.81 KDM4E (0.49) KDM4EHPGDMAPTCYP1A2CYP3A4
SCHEMBL25699196 0.81 CYP19A1 (0.50) KDM4EMEN1KMT2AHPGDMAPT
SCHEMBL3527999 0.81 CYP11B2 (0.45) KDM4EMEN1KMT2AHPGDCYP1A2
SCHEMBL24225402 0.79 TRPV4 (0.56) KDM4EMEN1KMT2AHPGDALDH1A1
SCHEMBL2954914 0.78 ALDH1A1 (0.56) KDM4EMEN1KMT2AHPGDMAPT
SCHEMBL10705073 0.77 AHR (0.43) KDM4EMEN1KMT2AHPGDMAPT
SCHEMBL27514116 0.76 KDM4E (0.49) KDM4EMEN1KMT2AHPGDMAPT
SCHEMBL24963528 0.76 PTGS2 (0.55) MEN1KMT2AMAPTALDH1A1MAOA
SCHEMBL25699199 0.76 CYP11B2 (0.40) KDM4EMEN1KMT2AHPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7759366-B2 Arylaminoaryl-alkyl-substituted imidazolidine-2,4-diones, process for preparing them, medicaments comprising these compounds, and their use SANOFI-AVENTIS (FR) 2010-07-20 US disclosed
US-20090215728-A1 Arylaminoaryl-alkyl-substituted imidazolidine-2,4-diones, process for preparing them, medicaments comprising these compounds, and their use SANOFI-AVENTIS (FR) 2009-08-27 US disclosed
EP-2061767-A1 ARYLAMINOARYL-ALKYL-SUBSTITUTED IMIDAZOLIDINE-2,4-DIONES, PROCESSES FOR PREPARING THEM, MEDICAMENTS COMPRISING THESE COMPOUNDS, AND THEIR USE Sanofi-Aventis (FR) 2009-05-27 EP disclosed
WO-2008017381-A1 ARYLAMINOARYL-ALKYL-SUBSTITUTED IMIDAZOLIDINE-2,4-DIONES, PROCESSES FOR PREPARING THEM, MEDICAMENTS COMPRISING THESE COMPOUNDS, AND THEIR USE SANOFI-AVENTIS (FR) 2008-02-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090215728-A1 Arylaminoaryl-alkyl-substituted imidazolidine-2,4-diones, process for preparing them, medicaments comprising these compounds, and their use GPR119, GIPR, LIPC KDM4E 477/4885MEN1 3627/4885KMT2A 1972/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.