SCHEMBL356138

SCHEMBL356138

CC(C)(C)OC(=O)N1CCCC1c1csc(N)n1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SCN4A P35499 1/20 0.45
USP30 Q70CQ3 5/20 0.45
UCHL1 P09936 3/20 0.45
HSD17B10 Q99714 1/20 0.45
ALDH1A1 P00352 3/20 0.44
SCN5A Q14524 1/20 0.43
SCN3A Q9NY46 1/20 0.43
ADAM17 P78536 2/20 0.43
L3MBTL1 Q9Y468 2/20 0.41
TSHR P16473 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
NPC1 O15118 1/20 0.40
LMNA P02545 1/20 0.40
HSD11B1 P28845 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8215613 1.00 SCN4A (0.45) SCN4AUSP30UCHL1HSD17B10ALDH1A1
SCHEMBL8240664 1.00 SCN4A (0.45) SCN4AUSP30UCHL1HSD17B10ALDH1A1
SCHEMBL29129342 0.86 USP30 (0.48) USP30UCHL1HSD17B10ALDH1A1L3MBTL1
SCHEMBL8218887 0.83 ADAM17 (0.46) SCN4AUSP30UCHL1ALDH1A1ADAM17
SCHEMBL354309 0.82 HSD17B10 (0.50) HSD17B10ALDH1A1ADAM17
SCHEMBL8222820 0.81 USP30 (0.51) USP30UCHL1ALDH1A1L3MBTL1TSHR
SCHEMBL23705673 0.81 TRPV3 (0.46) USP30HSD17B10ALDH1A1MEN1KMT2A
SCHEMBL8221844 0.81 USP30 (0.52) USP30UCHL1ALDH1A1L3MBTL1TSHR
SCHEMBL6468249 0.80 HSD11B1 (0.45) USP30UCHL1ALDH1A1L3MBTL1TSHR
SCHEMBL3060679 0.79 KDM4E (0.48) USP30ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117279896-A Amino substituted pyrido ring compounds, preparation method and application thereof 劲方医药科技(上海)有限公司 2023-12-22 CN disclosed
WO-2022214044-A1 AMINE-SUBSTITUTED PYRIDINE FUSED RING COMPOUNDS, PREPARATION METHOD THEREFOR AND USE THEREOF 劲方医药科技(上海)有限公司 2022-10-13 WO disclosed
EP-2200440-B1 ANTIBACTERIAL AMIDE AND SULFONAMIDE SUBSTITUTED HETEROCYCLIC UREA COMPOUNDS CRESTONE INC (US) 2017-07-19 EP disclosed
US-8148380-B2 Antibacterial amide and sulfonamide substituted heterocyclic urea compounds CRESTONE, INC. (US) 2012-04-03 US disclosed
US-20120015941-A1 Antibacterial Amide and Sulfonamide Substituted Heterocyclic Urea Compounds CRESTONE, INC. (US) 2012-01-19 US disclosed
EP-2200440-A1 ANTIBACTERIAL AMIDE AND SULFONAMIDE SUBSTITUTED HETEROCYCLIC UREA COMPOUNDS Crestone, Inc. (US) 2010-06-30 EP disclosed
WO-2009015208-A1 ANTIBACTERIAL AMIDE AND SULFONAMIDE SUBSTITUTED HETEROCYCLIC UREA COMPOUNDS REPLIDYNE, INC. (US) 2009-01-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120015941-A1 Antibacterial Amide and Sulfonamide Substituted Heterocyclic Urea Compounds NAAA, AADAC, RPSA SCN4A 1087/4885USP30 607/4885UCHL1 1492/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.