Indomethacin

Indomethacin

SCHEMBL356273

COc1ccc2c(c1)c(CC(=O)O)c(C)n2C(=O)c1ccc(Cl)cc1.COc1ccc2cc([C@H](C)C(=O)O)ccc2c1

nearest known ligand 0.79

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

PTGS1PTGS2

The experimentally established mechanism targets of Indomethacin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 known ✓ P35354 10/20 0.79
PTGS1 known ✓ P23219 3/20 0.79
AKR1C3 P42330 7/20 0.79
AKR1C2 P52895 6/20 0.79
HIF1A Q16665 3/20 0.79
ABCB1 P08183 2/20 0.79
GLO1 Q04760 2/20 0.79
AKR1C4 P17516 2/20 0.79
AKR1C1 Q04828 2/20 0.79
LMNA P02545 2/20 0.79
CYP1A2 P05177 2/20 0.79
CYP2D6 P10635 2/20 0.79
CYP2C9 P11712 2/20 0.79
NPSR1 Q6W5P4 2/20 0.79
KDM4E B2RXH2 1/20 0.79
MEN1 O00255 1/20 0.79
PTGES O14684 1/20 0.79
ABCC3 O15438 1/20 0.79
ABCC4 O15439 1/20 0.79
ABCB11 O95342 1/20 0.79

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Indomethacin SCHEMBL11570993 1.00 PTGS2 (0.79) PTGS2AKR1C3AKR1C2PTGS1HIF1A
Indomethacin SCHEMBL1307338 0.92 PTGS2 (0.75) PTGS2AKR1C3AKR1C2PTGS1HIF1A
Indomethacin SCHEMBL4300161 0.90 PTGS2 (0.74) PTGS2AKR1C3AKR1C2PTGS1HIF1A
Indomethacin SCHEMBL29525957 0.89 PTGS2 (1.00) PTGS2AKR1C3AKR1C2PTGS1HIF1A
Indomethacin SCHEMBL29353712 0.89 PTGS2 (1.00) PTGS2AKR1C3AKR1C2PTGS1HIF1A
Indomethacin SCHEMBL3518614 0.89 PTGS2 (1.00) PTGS2AKR1C3AKR1C2PTGS1HIF1A
Indomethacin SCHEMBL9300 0.89 PTGS2 (1.00) PTGS2AKR1C3AKR1C2PTGS1HIF1A
Indomethacin SCHEMBL23391006 0.88 PTGS2 (0.98) PTGS2AKR1C3AKR1C2PTGS1HIF1A
Indomethacin SCHEMBL8352438 0.88 PTGS2 (0.98) PTGS2AKR1C3AKR1C2PTGS1HIF1A
Indomethacin SCHEMBL1817813 0.88 PTGS2 (0.98) PTGS2AKR1C3AKR1C2PTGS1HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 60 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0278977-A1 PRODRUG DERIVATIVES OF CARBOXYLIC ACID DRUGS. BUNDGAARD HANS (DK) 1988-08-24 EP claimed
WO-1988001615-A1 PRODRUG DERIVATIVES OF CARBOXYLIC ACID DRUGS BUNDGAARD HANS (DK) 1988-03-10 WO claimed
US-12016764-B2 Tubular implants with controlled biodegradation POLY-MED, INC. (US) 2024-06-25 US disclosed
CN-111511310-B Tubular implant with controlled biodegradation 聚合-医药有限公司 2023-11-28 CN disclosed
US-20230255741-A1 MEDICAL IMPLANTS HAVING MANAGED BIODEGRADATION POLY-MED, INC. 2023-08-17 US disclosed
EP-3979947-A1 METHODS, DEVICES AND COMPOSITIONS FOR LOCAL DELIVERY Poly-Med Inc. (US) 2022-04-13 EP disclosed
US-20220071756-A1 TUBULAR IMPLANTS WITH CONTROLLED BIODEGRADATION POLY-MED, INC. 2022-03-10 US disclosed
CN-114096213-A Methods, devices and compositions for topical delivery 聚合-医药有限公司 2022-02-25 CN disclosed
CN-109414331-B Medical implant with managed biodegradation 聚合-医药有限公司 2021-09-21 CN disclosed
EP-3752201-A1 SUSPENSION OF NANOSCALE, ORGANIC PARTICLES AND PROCESS FOR PRODUCTION THEREOF Friedrich-Alexander-Universität Erlangen-Nürnberg (DE) 2020-12-23 EP disclosed
WO-2020252077-A1 METHODS, DEVICES AND COMPOSITIONS FOR LOCAL DELIVERY POLY-MED, INC. (US) 2020-12-17 WO disclosed
US-20090169471-A1 PARTICLES FOR INJECTION AND PROCESSES FOR FORMING THE SAME BOSTON SCIENTIFIC SCIMED, INC. (US) 2009-07-02 US disclosed
US-20090117039-A1 CHARGED BIODEGRADABLE POLYMERS FOR MEDICAL APPLICATIONS BOSTON SCIENTIFIC SCIMED, INC. (US) 2009-05-07 US disclosed
US-20090092677-A1 MULTI-COMPONENT PARTICLES FOR INJECTION AND PROCESSES FOR FORMING THE SAME BOSTON SCIENTIFIC SCIMED, INC. (US) 2009-04-09 US disclosed
US-20090053276-A1 INJECTABLE HYDROGEL COMPOSITIONS BOSTON SCIENTIFIC SCIMED, INC. (US) 2009-02-26 US disclosed
WO-2008115543-A2 UROLOGICAL MEDICAL DEVICES FOR RELEASE OF THERAPEUTIC AGENTS BOSTON SCIENTIFIC SCIMED, INC. (US) 2008-09-25 WO disclosed
US-20080234659-A1 UROLOGICAL MEDICAL DEVICES FOR RELEASE OF THERAPEUTIC AGENTS BOSTON SCIENTIFIC SCIMED, INC. (US) 2008-09-25 US disclosed
US-20080233167-A1 UROLOGICAL MEDICAL DEVICES FOR RELEASE OF PROSTATICALLY BENEFICIAL THERAPEUTIC AGENTS BOSTON SCIENTIFIC SCIMED, INC. (US) 2008-09-25 US disclosed
WO-2008115536-A2 UROLOGICAL MEDICAL DEVICES FOR RELEASE OF PROSTATICALLY BENEFICIAL THERAPEUTIC AGENTS BOSTON SCIENTIFIC SCIMED, INC. (US) 2008-09-25 WO disclosed
WO-1989008119-A1 HIGH MOLECULAR WEIGHT PRODRUG DERIVATIVES OF ANTI-INFLAMMATORY DRUGS SELCH LARSEN CLAUS (DK) 1989-09-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090053276-A1 INJECTABLE HYDROGEL COMPOSITIONS DLST, MPST, USP1 PTGS2 1651/4885PTGS1 1030/4885AKR1C3 4371/4885
US-20090169471-A1 PARTICLES FOR INJECTION AND PROCESSES FOR FORMING THE SAME LPXN, PGF, NUP205 PTGS2 384/4885PTGS1 285/4885AKR1C3 2788/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.