SCHEMBL3576804

SCHEMBL3576804

CNc1ncc(Cl)cc1C(=O)N(CCc1ccc(Cl)c(Cl)c1)Cc1ccc(C2CCCC2)cc1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 11/20 0.36
ALDH1A1 P00352 2/20 0.36
OPRK1 P41145 2/20 0.36
MAPT P10636 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
TSHR P16473 1/20 0.36
CYP2C19 P33261 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
MCHR1 Q99705 1/20 0.33
FFAR4 Q5NUL3 2/20 0.33
PROKR1 Q8TCW9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3576351 0.98 MCHR1 (0.35) SIGMAR1ALDH1A1OPRK1MAPTSMN1; SMN2
SCHEMBL3578672 0.90 GBA1 (0.34) SIGMAR1ALDH1A1OPRK1MAPTSMN1; SMN2
SCHEMBL3577036 0.89 MCHR1 (0.43) SIGMAR1ALDH1A1OPRK1MAPTSMN1; SMN2
SCHEMBL3583638 0.88 C5AR1 (0.41) MAPTOPRM1OPRD1MCHR1FFAR4
SCHEMBL3573512 0.85 HDAC1 (0.36) SIGMAR1CYP3A4TSHROPRM1OPRD1
SCHEMBL3574398 0.85 STAT3 (0.37) SMN1; SMN2CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL3576692 0.84 ESRRG (0.37) SIGMAR1OPRM1OPRD1
SCHEMBL3584245 0.83 SIGMAR1 (0.34) SIGMAR1ALDH1A1OPRK1MAPTSMN1; SMN2
SCHEMBL3573226 0.83 CNR1 (0.37) SMN1; SMN2CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL3574238 0.82 MLYCD (0.35) SIGMAR1CYP2C19OPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7678818-B2 Anthranilamide and 2-amino-heteroarene-carboxamide compounds HOFFMANN-LA ROCHE INC. (US) 2010-03-16 US claimed
EP-1984340-B1 ANTHRANILAMIDE/2-AMINO-HETEROARENE CARBOXAMIDE DERIVATIVES HOFFMANN LA ROCHE (CH) 2012-06-27 EP disclosed