SCHEMBL3583048

SCHEMBL3583048

Nc1cccc(NC(=O)OCc2ccccc2)c1

nearest known ligand 0.72

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 3/20 0.72
ENPP2 Q13822 3/20 0.64
BLK P51451 1/20 0.60
BTK Q06187 1/20 0.60
POLB P06746 1/20 0.58
TP53 P04637 2/20 0.56
MAPT P10636 2/20 0.56
NPC1 O15118 1/20 0.56
ALDH1A1 P00352 1/20 0.56
TSHR P16473 1/20 0.56
RAB9A P51151 1/20 0.56
ATM Q13315 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
DDX3X O00571 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3794371 0.92 MGLL (0.82) MGLLENPP2BLKBTKPOLB
SCHEMBL4577453 0.90 MGLL (0.65) MGLLENPP2BLKBTKPOLB
SCHEMBL3790408 0.87 MGLL (0.70) MGLLENPP2BLKBTKPOLB
SCHEMBL3789318 0.85 MGLL (0.85) MGLLENPP2POLBTP53MAPT
SCHEMBL3787599 0.85 MGLL (0.71) MGLLENPP2BLKBTKPOLB
SCHEMBL8984657 0.85 MGLL (0.76) MGLLENPP2POLBTP53MAPT
Benzyl Phenylcarbamate SCHEMBL1222943 0.84 POLB (0.78) MGLLENPP2POLBTP53MAPT
SCHEMBL3780622 0.84 MGLL (0.62) MGLLENPP2BLKBTKPOLB
SCHEMBL3784563 0.84 MGLL (0.62) MGLLENPP2BLKBTKPOLB
SCHEMBL27498433 0.84 MGLL (0.74) MGLLENPP2POLBTP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 41 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12404241-B2 Substituted 3-((3-aminophenyl)amino)piperidine-2,6-dione compounds, compositions thereof, and methods of treatment therewith CELGENE CORPORATION (US) 2025-09-02 US disclosed
US-20240368083-A1 SUBSTITUTED 3-((3-AMINOPHENYL)AMINO)PIPERIDINE-2,6-DIONE COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH CELGENE CORP (US) 2024-11-07 US disclosed
US-11873283-B2 Substituted 3-((3-aminophenyl)amino)piperidine-2,6-dione compounds, compositions thereof, and methods of treatment therewith CELGENE CORPORATION (US) 2024-01-16 US disclosed
US-20230002321-A1 SUBSTITUTED 3-((3-AMINOPHENYL)AMINO)PIPERIDINE-2,6-DIONE COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH CELGENE CORP (US) 2023-01-05 US disclosed
CN-113453681-A Substituted 3- ((3-aminophenyl) amino) piperidine-2, 6-dione compounds, compositions thereof, and methods of treatment using the same 细胞基因公司 2021-09-28 CN disclosed
US-10787436-B2 Inhibitors of cyclin-dependent kinase 7 (CDK7) DANA-FARBER CANCER INSTITUTE, INC. (US) 2020-09-29 US disclosed
US-10787436-B2 Inhibitors of cyclin-dependent kinase 7 (CDK7) DANA-FARBER CANCER INSTITUTE, INC. (US) 2020-09-29 US disclosed
CN-105732636-B Heteroaromatic compounds and their use in medicine 广东东阳光药业有限公司 2020-04-21 CN disclosed
US-20190100511-A1 INHIBITORS OF CYCLIN-DEPENDENT KINASE 7 (CDK7) DANA-FARBER CANCER INSTITUTE, INC. (US) 2019-04-04 US disclosed
US-20190100511-A1 INHIBITORS OF CYCLIN-DEPENDENT KINASE 7 (CDK7) DANA-FARBER CANCER INSTITUTE, INC. (US) 2019-04-04 US disclosed
WO-2006093832-A2 AMIDE DERIVATIVES AS ION-CHANNEL LIGANDS AND PHARMACEUTICAL COMPOSITIONS AND METHODS OF USING THE SAME RENOVIS, INC. (US) 2006-09-08 WO disclosed
US-20060194801-A1 Amide derivatives as ion-channel ligands and pharmaceutical compositions and methods of using the same EVOTEC AG (DE) 2006-08-31 US disclosed
US-6605626-B2 Benzamide inhibitors of factor Xa ELI LILLY AND COMPANY 2003-08-12 US disclosed
US-20020120007-A1 Benzamide inhibitors of factor Xa BEIGHT DOUGLAS WADE (US) 2002-08-29 US disclosed
US-6355810-B1 TREATMENT AND PREVENTION OF HYPERCHOLESTEROLEMIA, HYPERLIPIDEMIA, ATHEROSCLEROSIS ADVANCED MEDICINE, INC. 2002-03-12 US disclosed
US-6313122-B1 AS INHIBITORS OF FACTOR XA AND ARE USED AS ANTICOAGULANTS IN MAMMALS ELI LILLY AND COMPANY 2001-11-06 US disclosed
EP-1083894-A1 MULTIBINDING INHIBITORS OF HMG-CoA REDUCTASE Advanced Medicine, Inc. (US) 2001-03-21 EP disclosed
WO-1999063994-A9 MULTIBINDING INHIBITORS OF HMG-CoA REDUCTASE ADVANCED MEDICINE INC (US) 2000-07-27 WO disclosed
WO-1999063994-A1 MULTIBINDING INHIBITORS OF HMG-CoA REDUCTASE ADVANCED MEDICINE, INC. (US) 1999-12-16 WO disclosed
EP-0651740-B1 AMINO ACID LINKED NITROGEN MUSTARD DERIVATIVES AND THEIR USE AS PRODRUGS IN THE TREATMENT OF TUMOURS ZENECA LTD (GB) 1998-10-21 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190100511-A1 INHIBITORS OF CYCLIN-DEPENDENT KINASE 7 (CDK7) CDK7, CDK9, CDK6 MGLL 3798/4885ENPP2 459/4885BLK 219/4885
US-20230002321-A1 SUBSTITUTED 3-((3-AMINOPHENYL)AMINO)PIPERIDINE-2,6-DIONE COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH AR, NR5A2, ESRRA MGLL 4467/4885ENPP2 3460/4885BLK 2177/4885
US-11873283-B2 Substituted 3-((3-aminophenyl)amino)piperidine-2,6-dione compounds, compositions thereof, and methods of treatment therewith AR, NR5A2, ESRRA MGLL 4467/4885ENPP2 3460/4885BLK 2177/4885
US-20240368083-A1 SUBSTITUTED 3-((3-AMINOPHENYL)AMINO)PIPERIDINE-2,6-DIONE COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH AR, NR5A2, ESRRA MGLL 4467/4885ENPP2 3460/4885BLK 2177/4885
US-20060194801-A1 Amide derivatives as ion-channel ligands and pharmaceutical compositions and methods of using the same TRPV1, TRPA1, TRPV2 MGLL 1299/4885ENPP2 261/4885BLK 2185/4885
US-20020120007-A1 Benzamide inhibitors of factor Xa TFPI, F11, F12 MGLL 1026/4885ENPP2 330/4885BLK 1663/4885
US-12404241-B2 Substituted 3-((3-aminophenyl)amino)piperidine-2,6-dione compounds, compositions thereof, and methods of treatment therewith AR, NR5A2, ESRRA MGLL 4467/4885ENPP2 3460/4885BLK 2177/4885
US-10787436-B2 Inhibitors of cyclin-dependent kinase 7 (CDK7) CDK7, CDK9, CDK6 MGLL 3798/4885ENPP2 459/4885BLK 219/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.