SCHEMBL3583634

SCHEMBL3583634

CNc1ccc(Cl)cc1C(=O)N(CCc1ccc(F)c(Cl)c1)Cc1ccc(C(C)(C)C)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SERPINE1 P05121 1/20 0.39
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
GLA P06280 1/20 0.38
GAA P10253 1/20 0.38
NR1H4 Q96RI1 1/20 0.37
CCR9 P51686 2/20 0.37
CCR2 P41597 1/20 0.37
LMNA P02545 1/20 0.37
HTT P42858 1/20 0.37
KCNH2 Q12809 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
ESRRG P62508 3/20 0.37
ESRRB O95718 1/20 0.37
C5AR1 P21730 1/20 0.37
CNR2 P34972 1/20 0.36
FLT1 P17948 1/20 0.36
FLT4 P35916 1/20 0.36
KDR P35968 1/20 0.36
TP53 P04637 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3579634 0.92 SERPINE1 (0.40) SERPINE1KDM4EALDH1A1GLAGAA
SCHEMBL3570707 0.91 C5AR1 (0.39) KDM4EALDH1A1GLAGAANR1H4
SCHEMBL3584396 0.90 C5AR1 (0.44) SERPINE1KDM4EALDH1A1GLAGAA
SCHEMBL3575609 0.86 LMNA (0.43) SERPINE1LMNASMN1; SMN2C5AR1MEN1
SCHEMBL3581193 0.86 CCR9 (0.39) SERPINE1KDM4EALDH1A1GLAGAA
SCHEMBL3580741 0.86 C5AR1 (0.40) SERPINE1KDM4EALDH1A1GLAGAA
SCHEMBL3569982 0.83 LPAR1 (0.41) SERPINE1ALDH1A1GAANR1H4CCR9
SCHEMBL3580698 0.83 C5AR1 (0.44) KDM4EALDH1A1GLAGAACCR9
SCHEMBL3578799 0.83 TP53 (0.39) NR1H4ESRRGESRRBC5AR1TP53
SCHEMBL3577656 0.83 CNR1 (0.42) SERPINE1KDM4EALDH1A1GLAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7678818-B2 Anthranilamide and 2-amino-heteroarene-carboxamide compounds HOFFMANN-LA ROCHE INC. (US) 2010-03-16 US claimed
EP-1984340-B1 ANTHRANILAMIDE/2-AMINO-HETEROARENE CARBOXAMIDE DERIVATIVES HOFFMANN LA ROCHE (CH) 2012-06-27 EP disclosed