SCHEMBL3603373

SCHEMBL3603373

O=C(Cc1csc(N(Cc2cccnc2)C(=O)O)n1)N1CCOCC1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.46
MAPT P10636 3/20 0.46
HPGD P15428 1/20 0.46
GSTO1 P78417 2/20 0.46
KDM4E B2RXH2 1/20 0.42
POLB P06746 3/20 0.41
HSD11B1 P28845 1/20 0.40
FNTA P49354 1/20 0.39
FNTB P49356 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
FKBP1A P62942 1/20 0.39
LMNA P02545 6/20 0.38
TP53 P04637 5/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3615351 0.90 GSTO1 (0.47) ALDH1A1MAPTGSTO1KDM4EPOLB
SCHEMBL3604447 0.84 GSTO1 (0.42) ALDH1A1MAPTGSTO1KDM4EPOLB
SCHEMBL3600139 0.79 GSTO1 (0.52) MAPTGSTO1KDM4EPOLBMEN1
SCHEMBL3610003 0.79 GSTO1 (0.53) MAPTGSTO1POLBMEN1KMT2A
SCHEMBL3614294 0.78 GSTO1 (0.50) ALDH1A1MAPTGSTO1POLBMEN1
SCHEMBL3602399 0.75 GSTO1 (0.50) MAPTGSTO1POLBLMNATP53
SCHEMBL5599981 0.75 HSD11B1 (0.46) ALDH1A1MAPTHPGDHSD11B1MEN1
SCHEMBL3607138 0.75 SIGMAR1 (0.65)
SCHEMBL3601049 0.73 GSTO1 (0.48) ALDH1A1MAPTGSTO1POLBLMNA
SCHEMBL3609508 0.72 GSTO1 (0.47) ALDH1A1MAPTGSTO1POLBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100152188-A1 Novel Heterocyclic Compounds ORCHID RESEARCH LABORATORIES LIMITED (IN) 2010-06-17 US claimed
EP-2176229-B1 NOVEL CRYSTALLINE FORM OF 3-(DIFLUORMETHYL)-1-METHYL-N -(3',4',5'-TRIFLUOR[1,1'-BIPHENYL]-2-YL)-1H-PYRAZOL-4-CARBOXAMIDE BASF SE (DE) 2013-10-09 EP disclosed
US-20100160311-A1 Fungicidal Azolopyrimidines, Process for Their Preparation and Their Use For Controlling Harmful Fungi, and Also Compositions Comprising Them BASF SE (DE) 2010-06-24 US disclosed
US-20100152188-A1 Novel Heterocyclic Compounds ORCHID RESEARCH LABORATORIES LIMITED (IN) 2010-06-17 US disclosed
EP-2176229-A1 NOVEL CRYSTALLINE FORM OF 3-(DIFLUORMETHYL)-1-METHYL-N -(3',4',5'-TRIFLUOR[1,1'-BIPHENYL]-2-YL)-1H-PYRAZOL-4-CARBOXAMIDE BASF SE (DE) 2010-04-21 EP disclosed
EP-2057150-A1 THIOPHENE-SULFONIC ACID PICOLYL AMIDES BASF SE (DE) 2009-05-13 EP disclosed
WO-2009007344-A1 NOVEL CRYSTALLINE FORM OF 3-(DIFLUORMETHYL)-1-METHYL-N -(3',4',5'-TRIFLUOR[1,1'-BIPHENYL]-2-YL)-1H-PYRAZOL-4-CARBOXAMIDE BASF SE (DE) 2009-01-15 WO disclosed
WO-2008107398-A2 PYRAZINE COMPOUNDS BASF SE (DE) 2008-09-12 WO disclosed
WO-2008022937-A1 THIOPHENE-SULFONIC ACID PICOLYL AMIDES BASF SE (DE) 2008-02-28 WO disclosed
WO-2007017728-A2 NOVEL HETEROCYCLIC COMPOUNDS ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-02-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100160311-A1 Fungicidal Azolopyrimidines, Process for Their Preparation and Their Use For Controlling Harmful Fungi, and Also Compositions Comprising Them G6PD, CYP51A1, ERG28 ALDH1A1 912/4885MAPT 1401/4885HPGD 1757/4885
US-20100152188-A1 Novel Heterocyclic Compounds CYP11B2, CYP3A5, CYP11B1 ALDH1A1 370/4885MAPT 2986/4885HPGD 562/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.