SCHEMBL363897

SCHEMBL363897

CC(=O)C(c1ccccc1)(c1ccc(Br)cc1)c1ccnc(Cl)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.36
TLR7 Q9NYK1 1/20 0.35
KCNN4 O15554 3/20 0.34
TRPA1 O75762 1/20 0.34
MEN1 O00255 4/20 0.33
KMT2A Q03164 4/20 0.33
SMARCA2 P51531 2/20 0.33
SMARCA4 P51532 2/20 0.33
KDM5A P29375 1/20 0.33
KDM4C Q9H3R0 1/20 0.33
KDM5B Q9UGL1 1/20 0.33
KIF11 P52732 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
MAOB P27338 3/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
NR1H2 P55055 1/20 0.33
NR1H3 Q13133 1/20 0.33
NPC1 O15118 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL361971 0.85 NR1H2 (0.37) KCNN4MEN1KMT2AKIF11SMN1; SMN2
SCHEMBL364097 0.85 TRPA1 (0.35) ARTRPA1
SCHEMBL364575 0.76 KCNN4 (0.40) ARKCNN4SMARCA2SMARCA4KDM4C
SCHEMBL364193 0.73 NPC1 (0.34) ARTLR7RXFP1SMN1; SMN2NPC1
SCHEMBL363211 0.73 NPC1 (0.34) ARTLR7RXFP1SMN1; SMN2NPC1
SCHEMBL363549 0.73 NPC1 (0.34) ARTLR7RXFP1SMN1; SMN2NPC1
SCHEMBL371147 0.72 SORT1 (0.34) MEN1KMT2AMAOBSMN1; SMN2NPC1
SCHEMBL364536 0.72 SORT1 (0.35) CYP1A2CYP3A4ALDH1A1
SCHEMBL10538155 0.71 KIF11 (0.46) KCNN4MEN1KMT2AKIF11MAOB
SCHEMBL362869 0.71 TRPV1 (0.38) TLR7MEN1KMT2ARXFP1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed