SCHEMBL362157

SCHEMBL362157

CC(=O)[C@](c1ccc(C2CN(S(C)(=O)=O)C2)cc1)(c1ccnc(C)c1)c1ccccc1C

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PROKR1 Q8TCW9 1/20 0.34
TLR8 Q9NR97 1/20 0.32
TLR7 Q9NYK1 1/20 0.32
NR1I2 O75469 1/20 0.32
RORC P51449 1/20 0.32
MAP3K12 Q12852 2/20 0.31
GPBAR1 Q8TDU6 1/20 0.30
MMP3 P08254 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL364963 0.90 GPBAR1 (0.32) PROKR1TLR8TLR7GPBAR1
SCHEMBL363509 0.87 PROKR1 (0.40) PROKR1TLR8TLR7MAP3K12
SCHEMBL364745 0.83 MAPK1 (0.34) PROKR1TLR8TLR7
SCHEMBL362899 0.81 TLR8 (0.40) PROKR1TLR8TLR7MAP3K12GPBAR1
SCHEMBL363020 0.81 ATR (0.35)
SCHEMBL368721 0.80 WNT3A (0.44) MMP3
SCHEMBL363070 0.79 ALDH1A1 (0.41) PROKR1TLR8TLR7
SCHEMBL363061 0.79 KCNN4 (0.34) GPBAR1
SCHEMBL362081 0.78 HSD17B1 (0.33)
SCHEMBL363549 0.77 NPC1 (0.34) TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed