SCHEMBL362369

SCHEMBL362369

C=Nc1c(C(F)(F)F)cc(C(F)(F)F)cc1C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CES2 O00748 3/20 0.41
PTPN5 P54829 2/20 0.34
CACNA1H O95180 2/20 0.33
CACNA1B Q00975 1/20 0.33
CACNA1C Q13936 1/20 0.33
AR P10275 2/20 0.32
P2RX1 P51575 1/20 0.32
GPR35 Q9HC97 1/20 0.31
ALDH1A1 P00352 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C19 P33261 1/20 0.31
MAPT P10636 2/20 0.31
XBP1 P17861 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
PDE2A O00408 1/20 0.31
ITGB3 P05106 1/20 0.31
ITGAV P06756 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL364041 0.81 IDO1 (0.33)
SCHEMBL3175001 0.80 CES2 (0.43) CES2CACNA1HCACNA1BCACNA1CAR
SCHEMBL364195 0.79 RAC1 (0.35) ARALDH1A1CYP1A2CYP3A4CYP2C19
SCHEMBL12654823 0.74 TRPV4 (0.41) ARALDH1A1
SCHEMBL3190807 0.72 CES2 (0.40) CES2CACNA1HCACNA1BCACNA1CAR
SCHEMBL16488279 0.71 CES2 (0.46) CES2PTPN5ALDH1A1CYP3A4MAPT
SCHEMBL11603910 0.71 CES2 (0.43) CES2CACNA1HCACNA1BCACNA1CAR
SCHEMBL21851641 0.70 ITGB3 (0.45) CES2ALDH1A1MAPTITGB3ITGAV
SCHEMBL15933661 0.69 CES2 (0.41) CES2CACNA1HCACNA1BCACNA1CAR
SCHEMBL6756054 0.69 CES2 (0.41) CES2CACNA1HCACNA1BCACNA1CAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2311112-B1 ELECTRONIC DEVICES COMPRISING METAL COMPLEXES HAVING ISONITRILE LIGANDS MERCK PATENT GMBH (DE) 2012-03-14 EP disclosed
US-20110101327-A1 Electronic Devices Comprising Metal Complexes Having Isonitrile Ligands MERCK PATENT GMBH (DE) 2011-05-05 US disclosed
WO-2010015307-A1 ELECTRONIC DEVICES COMPRISING METAL COMPLEXES HAVING ISONITRILE LIGANDS MERCK PATENT GMBH (DE) 2010-02-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110101327-A1 Electronic Devices Comprising Metal Complexes Having Isonitrile Ligands EXOC4, ICMT, NCLN CES2 2721/4885PTPN5 2257/4885CACNA1H 521/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.