SCHEMBL363191

SCHEMBL363191

CC(=O)Nc1cccc(C(C/C(=N\O)c2c[nH]c(=O)c(C)c2)c2ccc(Cl)cc2F)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.38
MAPT P10636 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
POLB P06746 1/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
BRD4 O60885 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
CYP3A4 P08684 2/20 0.34
CYP2D6 P10635 2/20 0.34
SLC6A2 P23975 2/20 0.34
SLC6A4 P31645 2/20 0.34
SLC6A3 Q01959 2/20 0.34
KCNH2 Q12809 2/20 0.34
HPGD P15428 1/20 0.34
NPC1 O15118 1/20 0.33
PNP P00491 1/20 0.33
PARP1 P09874 1/20 0.33
SCN8A Q9UQD0 1/20 0.33
SCN10A Q9Y5Y9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL364598 0.90 ALDH1A1 (0.38) ALDH1A1MAPTMEN1KMT2APOLB
SCHEMBL363696 0.83 BRD4 (0.36) ALDH1A1MEN1KMT2ABRD4CYP2D6
SCHEMBL368193 0.81 CREBBP (0.40) ALDH1A1MAPTMEN1KMT2APOLB
SCHEMBL368191 0.81 CREBBP (0.40) ALDH1A1MAPTMEN1KMT2APOLB
SCHEMBL368192 0.81 CREBBP (0.40) ALDH1A1MAPTMEN1KMT2APOLB
SCHEMBL362423 0.81 BRD4 (0.35) MAPTBRD4CYP3A4CYP2D6PNP
SCHEMBL361680 0.81 GPBAR1 (0.47) POLBBRD4SLC6A3S1PR1S1PR3
SCHEMBL362797 0.79 GCGR (0.39) ALDH1A1POLBBRD4SLC6A3HPGD
SCHEMBL364696 0.79 GPBAR1 (0.38) BRD4S1PR1S1PR3
SCHEMBL362367 0.79 GPBAR1 (0.38) BRD4S1PR1S1PR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed