SCHEMBL362423

SCHEMBL362423

Cc1cc(/C(CC(c2cccc(C(=O)N(C)CCO)c2)c2ccc(Cl)cc2F)=N/O)c[nH]c1=O

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.35
PNP P00491 4/20 0.34
HCRTR1 O43613 1/20 0.33
MAPT P10636 1/20 0.31
PIK3CB P42338 2/20 0.31
GYS1 P13807 1/20 0.31
PIK3CA P42336 1/20 0.31
CDK4 P11802 1/20 0.31
CCND1 P24385 1/20 0.31
GPBAR1 Q8TDU6 1/20 0.31
LMNA P02545 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
HTT P42858 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL363696 0.85 BRD4 (0.36) BRD4PNPCYP1A2CYP2D6CYP2C9
SCHEMBL369844 0.82 BRD4 (0.33) BRD4PIK3CBGYS1PIK3CALMNA
SCHEMBL369842 0.82 BRD4 (0.33) BRD4PIK3CBGYS1PIK3CALMNA
SCHEMBL369843 0.82 BRD4 (0.33) BRD4PIK3CBGYS1PIK3CALMNA
SCHEMBL363191 0.81 ALDH1A1 (0.38) BRD4PNPMAPTCYP3A4CYP2D6
SCHEMBL361680 0.78 GPBAR1 (0.47) BRD4GPBAR1
SCHEMBL364494 0.78 GPBAR1 (0.47) BRD4HCRTR1CDK4CCND1GPBAR1
SCHEMBL362797 0.78 GCGR (0.39) BRD4GPBAR1
SCHEMBL363638 0.77 GPBAR1 (0.41) GPBAR1
SCHEMBL363248 0.77 GPBAR1 (0.41) GPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed