SCHEMBL3637159

SCHEMBL3637159

COc1ccc(-c2csc(Nc3ccc(-c4nc(C)c[nH]4)c(OC)c3)n2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.60
MEN1 O00255 7/20 0.58
KMT2A Q03164 7/20 0.58
MAPT P10636 6/20 0.58
RAB9A P51151 5/20 0.58
GAA P10253 4/20 0.58
NPC1 O15118 4/20 0.58
SMN1; SMN2 Q16637 4/20 0.58
ALOX5 P09917 4/20 0.55
VCP P55072 1/20 0.54
NFKB1 P19838 3/20 0.54
NFKB2 Q00653 3/20 0.54
RELA Q04206 3/20 0.54
ALDH1A1 P00352 3/20 0.54
MCL1 Q07820 1/20 0.54
RECQL P46063 1/20 0.54
MAPK1 P28482 1/20 0.53
TUBB4A P04350 1/20 0.53
TUBB P07437 1/20 0.53
TUBA3C P0DPH7 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3635139 0.91 ALOX5 (0.69) PTGS2MEN1KMT2AMAPTALOX5
SCHEMBL3641518 0.90 PTGS2 (0.56) PTGS2MEN1KMT2AMAPTRAB9A
SCHEMBL3637592 0.89 CSNK2A1 (0.53) PTGS2MEN1KMT2AMAPTGAA
SCHEMBL3634967 0.86 ALOX5 (0.55) PTGS2MEN1KMT2AMAPTRAB9A
SCHEMBL3637805 0.85 VCP (0.59) PTGS2MEN1KMT2AMAPTGAA
SCHEMBL3640999 0.83 CYP1B1 (0.53) PTGS2MEN1KMT2AMAPTRAB9A
SCHEMBL3640612 0.83 AMY1A (0.54) PTGS2MAPTALOX5VCPALDH1A1
SCHEMBL3632755 0.83 ALOX5 (0.53) PTGS2MEN1KMT2AMAPTGAA
SCHEMBL3633219 0.83 PSEN1 (0.64) PTGS2MEN1KMT2AMAPTGAA
SCHEMBL1041244 0.83 CYP1A1 (0.53) PTGS2MEN1KMT2AMAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2155740-A1 HETARYLANILINES AS MODULATORS FOR AMYLOID BETA F. Hoffmann-Roche AG (CH) 2010-02-24 EP disclosed
WO-2008138753-A1 HETARYLANILINES AS MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2008-11-20 WO disclosed