SCHEMBL364494

SCHEMBL364494

Cc1ccccc1C(C/C(=N\O)c1c[nH]c(=O)c(C)c1)c1ccc(C(=O)N(C)CCO)cc1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 6/20 0.47
BRD4 O60885 1/20 0.40
HCRTR1 O43613 1/20 0.34
USP1 O94782 2/20 0.33
CDK4 P11802 5/20 0.33
CCND1 P24385 5/20 0.33
CDK2 P24941 2/20 0.32
HDAC6 Q9UBN7 1/20 0.32
PDK2 Q15119 1/20 0.32
MGAM O43451 2/20 0.32
GAA P10253 2/20 0.32
SI P14410 2/20 0.32
MGAM2 Q2M2H8 2/20 0.32
TACR1 P25103 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL361679 0.90 GPBAR1 (0.47) GPBAR1BRD4HCRTR1MGAMGAA
SCHEMBL363678 0.86 GPBAR1 (0.61) GPBAR1BRD4MGAMGAASI
SCHEMBL364601 0.83 GPBAR1 (0.66) GPBAR1BRD4MGAMGAASI
SCHEMBL362545 0.83 GPBAR1 (0.66) GPBAR1BRD4MGAMGAASI
SCHEMBL363349 0.83 GPBAR1 (0.66) GPBAR1BRD4MGAMGAASI
SCHEMBL364032 0.83 GPBAR1 (0.47) GPBAR1BRD4
SCHEMBL364092 0.82 GPBAR1 (0.48) GPBAR1BRD4MGAMGAASI
SCHEMBL1390451 0.81 GPBAR1 (0.48) GPBAR1BRD4USP1HDAC6
SCHEMBL1389724 0.81 GPBAR1 (0.71) GPBAR1USP1HDAC6PDK2
SCHEMBL364212 0.81 GPBAR1 (0.71) GPBAR1USP1HDAC6PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed