SCHEMBL364524

SCHEMBL364524

COCCNC(=O)c1ccc(C(C/C(=N\O)c2c[nH]c(=O)c(C)c2)c2ccccc2Cl)cc1F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.36
HAT1 O14929 2/20 0.35
EP300 Q09472 2/20 0.35
BRD4 O60885 1/20 0.35
ALDH1A1 P00352 4/20 0.34
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
PYGL P06737 1/20 0.34
POLB P06746 1/20 0.34
KDM4E B2RXH2 1/20 0.33
MAPT P10636 1/20 0.33
HTT P42858 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
GPBAR1 Q8TDU6 2/20 0.33
MAPK14 Q16539 1/20 0.33
TNKS2 Q9H2K2 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA3 P07451 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL364487 0.91 BRD4 (0.42) BRD4GPBAR1F9CTSA
SCHEMBL363071 0.89 BRD4 (0.37) BRD4GPBAR1F9CTSA
SCHEMBL361665 0.87 HPGD (0.37) BRD4POLBGPBAR1MAPK14HPGD
SCHEMBL362147 0.85 MET (0.34) HAT1EP300BRD4GPBAR1F9
SCHEMBL362599 0.85 BRD4 (0.40) EP300BRD4GPBAR1MAPK14HPGD
SCHEMBL363606 0.85 GPBAR1 (0.35) BRD4POLBGPBAR1MAPK14HPGD
SCHEMBL364618 0.84 MET (0.42) BRD4KDM4ENPSR1GPBAR1HPGD
SCHEMBL364504 0.83 GPBAR1 (0.40) BRD4NPC1KDM4EMAPTGPBAR1
SCHEMBL368843 0.83 ALDH1A1 (0.36) HAT1EP300BRD4ALDH1A1NPC1
SCHEMBL368841 0.83 ALDH1A1 (0.36) HAT1EP300BRD4ALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed