SCHEMBL3650322

SCHEMBL3650322

CNC(=O)OC(c1cc(-c2cccnc2F)c(S(=O)(=O)c2cccc(OC)c2)s1)C(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 4/20 0.38
GLO1 Q04760 1/20 0.37
SLC40A1 Q9NP59 1/20 0.37
ABCC9 O60706 1/20 0.37
ABCC8 Q09428 1/20 0.37
KCNJ11 Q14654 1/20 0.37
KCNJ8 Q15842 1/20 0.37
NPC1 O15118 1/20 0.37
MET P08581 1/20 0.35
GAA P10253 1/20 0.35
KAT6A Q92794 1/20 0.35
NAMPT P43490 4/20 0.34
MEP1B Q16820 1/20 0.33
MMP2 P08253 1/20 0.33
MMP9 P14780 1/20 0.33
MMP8 P22894 1/20 0.33
MMP13 P45452 1/20 0.33
PGAM1 P18669 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3653602 0.88 NAT1 (0.31) NAMPTALDH1A1
SCHEMBL3651480 0.87 ABCC9 (0.37) NFE2L2GLO1SLC40A1ABCC9ABCC8
SCHEMBL3654637 0.87 NR3C1 (0.38) GLO1SLC40A1KAT6ANAMPT
SCHEMBL3803807 0.86 ALDH1A1 (0.31) ALDH1A1
SCHEMBL3650372 0.83 NR3C1 (0.35) GLO1SLC40A1NAMPT
SCHEMBL3648322 0.82 ALDH1A1 (0.31) ALDH1A1
Hydrochloric Acid SCHEMBL3649192 0.81 NR3C1 (0.36) GLO1SLC40A1NAMPT
SCHEMBL3653610 0.81 PIK3CA (0.35) NPC1
SCHEMBL3652253 0.80 HTR6 (0.32)
SCHEMBL2409435 0.78 MET (0.43) NFE2L2GLO1SLC40A1ABCC9ABCC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed