SCHEMBL3650372

SCHEMBL3650372

CNC(=O)OC(c1cc(-c2cccnc2F)c(S(=O)(=O)c2cccc(Br)c2)s1)C(C)(C)C.CNC(=O)OC(c1cc(-c2cccnc2F)c(S(=O)(=O)c2cccc(C#N)c2)s1)C(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 1/20 0.35
GLO1 Q04760 1/20 0.33
SLC40A1 Q9NP59 1/20 0.33
NAMPT P43490 1/20 0.33
GRM5 P41594 1/20 0.32
APLNR P35414 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3654637 0.95 NR3C1 (0.38) NR3C1GLO1SLC40A1NAMPTGRM5
Hydrochloric Acid SCHEMBL3649192 0.89 NR3C1 (0.36) NR3C1GLO1SLC40A1NAMPTAPLNR
SCHEMBL3650322 0.83 NFE2L2 (0.38) GLO1SLC40A1NAMPT
SCHEMBL3653602 0.82 NAT1 (0.31) NAMPT
SCHEMBL3803807 0.81 ALDH1A1 (0.31)
SCHEMBL3652253 0.78 HTR6 (0.32)
Hydrochloric Acid SCHEMBL3650276 0.78 HTR6 (0.34)
SCHEMBL3648322 0.77 ALDH1A1 (0.31)
SCHEMBL3652075 0.75 LIPG (0.31)
SCHEMBL3647878 0.74 ABCC9 (0.38) NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed