SCHEMBL365034

SCHEMBL365034

CS(=O)(=O)NC(=O)c1ccc(OCc2cc(Cl)ccc2Cl)cc1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 11/20 0.54
SCN5A Q14524 2/20 0.54
NR4A2 P43354 1/20 0.51
MAOB P27338 2/20 0.47
BCL2L1 Q07817 2/20 0.47
MCL1 Q07820 2/20 0.47
HDAC8 Q9BY41 1/20 0.46
ADAMTS4 O75173 1/20 0.46
MMP1 P03956 1/20 0.46
MMP13 P45452 1/20 0.46
MAOA P21397 1/20 0.46
PTGER4 P35408 1/20 0.46
EPHX2 P34913 1/20 0.45
NR1H4 Q96RI1 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14890261 0.90 NR4A2 (0.64) SCN9ASCN5ANR4A2MAOBHDAC8
SCHEMBL14890406 0.87 ALDH1A1 (0.53) SCN9ASCN5AMCL1HDAC8PTGER4
SCHEMBL14890410 0.86 SCN9A (0.57) SCN9ASCN5ANR4A2MAOBMMP1
SCHEMBL364245 0.85 MAOA (0.65) SCN9ASCN5ANR4A2MAOBBCL2L1
SCHEMBL365210 0.82 MAOA (0.63) SCN9ASCN5ANR4A2MAOBBCL2L1
SCHEMBL366081 0.82 MAOA (0.63) SCN9ASCN5ANR4A2MAOBBCL2L1
SCHEMBL10203178 0.81 SCN9A (0.66) SCN9ASCN5AMAOBBCL2L1MCL1
SCHEMBL367348 0.81 BCL2L1 (0.57) SCN9ASCN5ANR4A2MAOBBCL2L1
SCHEMBL366514 0.81 ADAMTS5 (0.59) SCN9ASCN5ANR4A2MAOBADAMTS4
SCHEMBL365474 0.81 MAOB (0.67) NR4A2MAOBBCL2L1MCL1ADAMTS4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9096500-B2 Acyl sulfonamide compounds PFIZER LIMITED (GB) 2015-08-04 US disclosed
EP-2593428-B1 N-SULFONYLBENZAMIDES AS INHIBITORS OF VOLTAGE-GATED SODIUM CHANNELS PFIZER LTD (GB) 2014-11-19 EP disclosed
EP-2593428-A2 N-SULFONYLBENZAMIDES AS INHIBITORS OF VOLTAGE-GATED SODIUM CHANNELS Pfizer Limited (GB) 2013-05-22 EP disclosed
US-20130109701-A1 Chemical Compounds PFIZER LIMITED (GB) 2013-05-02 US disclosed
WO-2012007868-A2 CHEMICAL COMPOUNDS PFIZER LIMITED (GB) 2012-01-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130109701-A1 Chemical Compounds SCN1A, SCN1B, SCN7A SCN9A 16/4885SCN5A 5/4885NR4A2 1933/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.