SCHEMBL365488

SCHEMBL365488

CC(=O)c1ccc2c(C(=O)N(C)CCN(C)C)c3ccccc3n2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 4/20 0.41
TNF P01375 2/20 0.39
ALDH1A1 P00352 2/20 0.38
HPGD P15428 1/20 0.38
EGFR P00533 2/20 0.37
SRC P12931 2/20 0.37
HDAC1 Q13547 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
CNR2 P34972 2/20 0.35
PRKCB P05771 1/20 0.35
PRKCA P17252 1/20 0.35
PRKCH P24723 1/20 0.35
PRKCQ Q04759 1/20 0.35
PRKCD Q05655 1/20 0.35
TNFSF11 O14788 1/20 0.35
POLR1A O95602 1/20 0.35
TACR1 P25103 1/20 0.35
HTR7 P34969 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL366300 0.88 CNR2 (0.38) PARP1TNFALDH1A1HPGDEGFR
SCHEMBL366186 0.84 ALDH1A1 (0.39) ALDH1A1HPGDEGFRSRCHDAC1
SCHEMBL364305 0.84 ALDH1A1 (0.36) ALDH1A1HPGDEGFRSRCHDAC1
SCHEMBL366838 0.81 ALDH1A1 (0.41) ALDH1A1HPGDEGFRSRCHDAC1
SCHEMBL365487 0.81 POLR1A (0.40) PARP1TNFALDH1A1HPGDPOLR1A
SCHEMBL366239 0.81 PLA2G2A (0.41) ALDH1A1HPGDCNR2PRKCBPRKCA
SCHEMBL364862 0.81 EGFR (0.56) ALDH1A1HPGDEGFRSRCHDAC1
SCHEMBL364892 0.81 ALDH1A1 (0.47) PARP1TNFALDH1A1
SCHEMBL367569 0.80 SRC (0.46) ALDH1A1HPGDEGFRSRC
SCHEMBL365762 0.80 ALDH1A1 (0.44) ALDH1A1HPGDUTS2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007007-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007007-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed