SCHEMBL366300

SCHEMBL366300

CC(=O)c1ccc2c(C(=S)N(C)CCN(C)C)c3ccccc3n2c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 2/20 0.38
HDAC1 Q13547 2/20 0.37
HDAC10 Q969S8 2/20 0.37
HDAC8 Q9BY41 2/20 0.37
HDAC6 Q9UBN7 2/20 0.37
PRKCA P17252 2/20 0.36
PRKCB P05771 1/20 0.36
PRKCH P24723 1/20 0.36
PRKCQ Q04759 1/20 0.36
PRKCD Q05655 1/20 0.36
ALDH1A1 P00352 2/20 0.36
HPGD P15428 1/20 0.36
HTR6 P50406 6/20 0.36
PARP1 P09874 2/20 0.36
EGFR P00533 1/20 0.35
SRC P12931 1/20 0.35
HTR2C P28335 2/20 0.34
HTR2A P28223 1/20 0.34
TNF P01375 1/20 0.34
HDAC3 O15379 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL365488 0.88 PARP1 (0.41) CNR2HDAC1HDAC10HDAC8HDAC6
SCHEMBL366186 0.82 ALDH1A1 (0.39) CNR2HDAC1HDAC10HDAC8HDAC6
SCHEMBL366455 0.82 EGFR (0.48) HDAC1HDAC10HDAC8HDAC6ALDH1A1
SCHEMBL366299 0.82 LMNA (0.38) CNR2ALDH1A1HPGDPARP1EGFR
SCHEMBL364305 0.82 ALDH1A1 (0.36) CNR2HDAC1HDAC10HDAC8HDAC6
SCHEMBL366838 0.80 ALDH1A1 (0.41) CNR2HDAC1HDAC10HDAC8HDAC6
SCHEMBL366239 0.80 PLA2G2A (0.41) CNR2PRKCAPRKCBPRKCHPRKCQ
SCHEMBL364862 0.80 EGFR (0.56) HDAC1HDAC10HDAC8HDAC6ALDH1A1
SCHEMBL367569 0.79 SRC (0.46) ALDH1A1HPGDEGFRSRC
SCHEMBL365762 0.78 ALDH1A1 (0.44) ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007007-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007007-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed