SCHEMBL366186

SCHEMBL366186

CC(=O)c1ccc2c(C(=O)CCN(C)C)c3ccccc3n2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.39
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
STAT6 P42226 1/20 0.39
HSD17B10 Q99714 1/20 0.39
EGFR P00533 4/20 0.38
HPGD P15428 1/20 0.38
GSR P00390 2/20 0.37
SRC P12931 2/20 0.37
PLA2G2A P14555 1/20 0.37
HDAC1 Q13547 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
LMNA P02545 1/20 0.36
PRNP P04156 1/20 0.36
CHRM2 P08172 1/20 0.36
HTR1A P08908 1/20 0.36
ADRA2A P08913 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL366239 0.92 PLA2G2A (0.41) ALDH1A1CYP1A2HPGDPLA2G2ALMNA
SCHEMBL366838 0.88 ALDH1A1 (0.41) ALDH1A1EGFRHPGDSRCPLA2G2A
SCHEMBL364305 0.87 ALDH1A1 (0.36) ALDH1A1EGFRHPGDSRCPLA2G2A
SCHEMBL365488 0.84 PARP1 (0.41) ALDH1A1EGFRHPGDSRCHDAC1
SCHEMBL367619 0.84 ALDH1A1 (0.39) ALDH1A1HPGDPLA2G2ACNR2
SCHEMBL366442 0.83 ALDH1A1 (0.42) ALDH1A1CYP1A2CYP3A4EGFRHPGD
SCHEMBL364862 0.82 EGFR (0.56) ALDH1A1CYP1A2HSD17B10EGFRHPGD
SCHEMBL366300 0.82 CNR2 (0.38) ALDH1A1EGFRHPGDSRCHDAC1
SCHEMBL364389 0.82 ALDH1A1 (0.48) ALDH1A1EGFRHPGDSRCLMNA
SCHEMBL365469 0.82 PLA2G2A (0.39) ALDH1A1HPGDPLA2G2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007007-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007007-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed