SCHEMBL366838

SCHEMBL366838

CC(=O)c1ccc2c(C(=O)CN(C)C)c3ccccc3n2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 1/20 0.41
USP2 O75604 1/20 0.41
HPGD P15428 1/20 0.40
NPY5R Q15761 1/20 0.36
EGFR P00533 4/20 0.36
SRC P12931 3/20 0.36
KMT2A Q03164 2/20 0.34
HDAC6 Q9UBN7 3/20 0.34
HDAC1 Q13547 2/20 0.34
HDAC10 Q969S8 2/20 0.34
HDAC8 Q9BY41 2/20 0.34
HDAC3 O15379 1/20 0.34
HDAC2 Q92769 1/20 0.34
NCOR2 Q9Y618 1/20 0.34
MEN1 O00255 1/20 0.34
CREBBP Q92793 2/20 0.34
CXCR3 P49682 1/20 0.34
PLA2G2A P14555 1/20 0.34
TSPO P30536 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL364305 0.89 ALDH1A1 (0.36) ALDH1A1HPGDEGFRSRCKMT2A
SCHEMBL367061 0.88 KDM4E (0.43) ALDH1A1KDM4EUSP2HPGDNPY5R
SCHEMBL366186 0.88 ALDH1A1 (0.39) ALDH1A1HPGDEGFRSRCKMT2A
SCHEMBL366442 0.85 ALDH1A1 (0.42) ALDH1A1KDM4EHPGDEGFRSRC
SCHEMBL366239 0.84 PLA2G2A (0.41) ALDH1A1HPGDKMT2AMEN1PLA2G2A
SCHEMBL364389 0.84 ALDH1A1 (0.48) ALDH1A1KDM4EHPGDEGFRSRC
SCHEMBL366194 0.84 CNR1 (0.35) ALDH1A1KDM4EHPGDEGFRSRC
SCHEMBL367569 0.83 SRC (0.46) ALDH1A1KDM4EHPGDEGFRSRC
SCHEMBL365488 0.81 PARP1 (0.41) ALDH1A1HPGDEGFRSRCHDAC6
SCHEMBL367619 0.81 ALDH1A1 (0.39) ALDH1A1HPGDPLA2G2ACNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007007-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007007-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed