SCHEMBL3656280

SCHEMBL3656280

COC(=O)c1cc(-c2nnn[nH]2)cc(-c2ncccc2OC)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.38
KDM4E B2RXH2 2/20 0.38
HTT P42858 2/20 0.38
ALOX15 P16050 1/20 0.38
MAPT P10636 2/20 0.37
HPGD P15428 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
CBFB Q13951 1/20 0.35
MAP2K1 Q02750 1/20 0.35
POLB P06746 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
PKM P14618 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
SMPD3 Q9NY59 1/20 0.34
NEK1 Q96PY6 1/20 0.34
CDK8 P49336 1/20 0.33
MAP2K4 P45985 1/20 0.33
GRM5 P41594 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3655146 0.90 CBFB (0.36) ALDH1A1KDM4EHTTL3MBTL1CBFB
SCHEMBL3655959 0.83 ADORA3 (0.42) ALDH1A1KDM4EALOX15MAPTHPGD
SCHEMBL733150 0.79 GABRG2 (0.44) ALDH1A1KDM4ESMN1; SMN2NEK1CDK8
SCHEMBL3800296 0.78 ROCK2 (0.39) ALDH1A1HTT
SCHEMBL2203896 0.78 ATAD2 (0.46) ALDH1A1KDM4EHTTALOX15MAPT
SCHEMBL3659131 0.76 HPGDS (0.39) ALDH1A1KDM4EMAPTPOLBCDK8
SCHEMBL3658350 0.76 MAPT (0.45) ALDH1A1KDM4EMAPTHPGDPOLB
SCHEMBL2512905 0.75 KDM4E (0.48) ALDH1A1KDM4EMAPTHPGDL3MBTL1
SCHEMBL1505455 0.75 GABRG2 (0.50) ALDH1A1MAPTHPGDNEK1CDK8
SCHEMBL2203174 0.73 TP53 (0.56) ALDH1A1MAPTHPGDL3MBTL1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2205573-A1 TETRAZOLE-SUBSTITUTED ARYL AMIDE DERIVATIVES AND USES THEREOF F. Hoffmann-Roche AG (CH) 2010-07-14 EP disclosed
WO-2009043780-A1 TETRAZOLE-SUBSTITUTED ARYL AMIDE DERIVATIVES AND USES THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2009-04-09 WO disclosed