SCHEMBL365647

SCHEMBL365647

NS(=O)(=O)c1ccc2c(C(=O)O)c3ccccn3c2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.43
PTGS2 P35354 1/20 0.42
EGFR P00533 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
STAT6 P42226 1/20 0.39
HIF1A Q16665 1/20 0.39
MAPT P10636 3/20 0.39
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
APAF1 O14727 1/20 0.39
G6PD P11413 1/20 0.39
PABPC1 P11940 1/20 0.39
CACNA1B Q00975 1/20 0.39
APBA1 Q02410 1/20 0.39
KMT2A Q03164 1/20 0.39
SAE1 Q9UBE0 1/20 0.39
UBA2 Q9UBT2 1/20 0.39
CA1 P00915 7/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL364652 0.90 CA2 (0.40) IDO1EGFRMAPTALDH1A1KDM4E
SCHEMBL367746 0.86 EGFR (0.43) IDO1PTGS2EGFRMAPTALDH1A1
SCHEMBL365426 0.85 MAPT (0.47) IDO1MAPTALDH1A1KDM4EMEN1
SCHEMBL366461 0.84 HTT (0.46) IDO1PTGS2EGFRMAPTALDH1A1
SCHEMBL365146 0.82 IDO1 (0.40) IDO1PTGS2EGFRMAPTALDH1A1
SCHEMBL366103 0.82 ALDH1A1 (0.60) IDO1CYP1A2CYP3A4HIF1AMAPT
SCHEMBL366810 0.79 PTGS2 (0.45) IDO1PTGS2EGFRCYP3A4MAPT
SCHEMBL365934 0.79 KDM4E (0.45) IDO1PTGS2EGFRMAPTALDH1A1
SCHEMBL366887 0.79 KDM4E (0.56) IDO1PTGS2EGFRMAPTALDH1A1
SCHEMBL366132 0.78 ALDH1A1 (0.38) IDO1PTGS2EGFRCYP1A2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed