SCHEMBL366132

SCHEMBL366132

CN(C)CCS(=O)(=O)c1ccc2c(C(=O)O)c3ccccn3c2c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.38
KDM4E B2RXH2 2/20 0.38
HSD17B10 Q99714 1/20 0.38
AGTR1 P30556 5/20 0.37
IDO1 P14902 3/20 0.37
HTR6 P50406 5/20 0.36
MEN1 O00255 1/20 0.36
APAF1 O14727 1/20 0.36
MAPT P10636 1/20 0.36
G6PD P11413 1/20 0.36
PABPC1 P11940 1/20 0.36
CACNA1B Q00975 1/20 0.36
APBA1 Q02410 1/20 0.36
KMT2A Q03164 1/20 0.36
SAE1 Q9UBE0 1/20 0.36
UBA2 Q9UBT2 1/20 0.36
PTGS2 P35354 1/20 0.36
CNR2 P34972 1/20 0.36
POLB P06746 2/20 0.36
CYP1A2 P05177 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL364605 0.90 HTR6 (0.37) ALDH1A1KDM4EHSD17B10AGTR1IDO1
SCHEMBL365521 0.88 KMT2A (0.43) ALDH1A1KDM4EHSD17B10IDO1MEN1
SCHEMBL366692 0.86 ALDH1A1 (0.43) ALDH1A1KDM4EHSD17B10IDO1HTR6
SCHEMBL366461 0.83 HTT (0.46) ALDH1A1KDM4EAGTR1IDO1MEN1
SCHEMBL366133 0.82 AGTR1 (0.41) AGTR1HTR6HTR1ADRD2HTR1D
SCHEMBL367746 0.81 EGFR (0.43) ALDH1A1KDM4EAGTR1IDO1MEN1
SCHEMBL365647 0.78 IDO1 (0.43) ALDH1A1KDM4EAGTR1IDO1MEN1
SCHEMBL366857 0.75 ALDH1A1 (0.44) ALDH1A1KDM4EHSD17B10IDO1MEN1
SCHEMBL366535 0.75 EGFR (0.48) ALDH1A1KDM4EHSD17B10IDO1MAPT
SCHEMBL365146 0.74 IDO1 (0.40) ALDH1A1KDM4EAGTR1IDO1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed