SCHEMBL366015

SCHEMBL366015

N#CCOc1cc(OCCc2cccnc2)c2c(C(N)=O)c3ccccn3c2c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 7/20 0.37
CYP11B2 P19099 7/20 0.37
CYP19A1 P11511 3/20 0.37
MKNK1 Q9BUB5 2/20 0.37
MKNK2 Q9HBH9 2/20 0.37
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
GRM2 Q14416 1/20 0.35
GCK P35557 1/20 0.33
MAPK12 P53778 1/20 0.33
MAPK14 Q16539 1/20 0.33
HSD17B10 Q99714 1/20 0.33
OPRM1 P35372 1/20 0.33
OPRK1 P41145 1/20 0.33
KCNH2 Q12809 1/20 0.33
JAK2 O60674 1/20 0.32
JAK1 P23458 1/20 0.32
PDE4A P27815 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL364642 0.92 CYP11B1 (0.40) CYP11B1CYP11B2CYP19A1MKNK1MKNK2
SCHEMBL365964 0.92 KDM4E (0.36) CYP11B1CYP11B2CYP19A1KDM4EALDH1A1
SCHEMBL364640 0.90 ALDH1A1 (0.39) KDM4EALDH1A1MEN1KMT2APDE4A
SCHEMBL366694 0.85 MKNK1 (0.41) CYP11B1CYP11B2CYP19A1MKNK1MKNK2
SCHEMBL367248 0.84 ALDH1A1 (0.37) KDM4EALDH1A1MEN1KMT2AHSD17B10
SCHEMBL365785 0.84 ALDH1A1 (0.38) KDM4EALDH1A1MEN1KMT2AOPRM1
SCHEMBL367193 0.84 GPR132 (0.38) KDM4EALDH1A1HSD17B10
SCHEMBL366072 0.83 FFAR1 (0.37) CYP11B1CYP11B2CYP19A1KDM4EALDH1A1
SCHEMBL366806 0.80 ALDH1A1 (0.35) KDM4EALDH1A1MEN1KMT2A
SCHEMBL367224 0.80 ALDH1A1 (0.43) MKNK2KDM4EALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed