SCHEMBL366455

SCHEMBL366455

CC(=O)c1ccc2c(C(=S)NCCN(C)C)c3ccccc3n2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.48
SRC P12931 1/20 0.48
KDM4E B2RXH2 3/20 0.42
MAPT P10636 2/20 0.42
HPGD P15428 3/20 0.41
ALDH1A1 P00352 3/20 0.41
HSD17B10 Q99714 1/20 0.41
ATM Q13315 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
FYN P06241 1/20 0.36
RAD52 P43351 1/20 0.36
CYP1A2 P05177 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
TP53 P04637 1/20 0.36
IDO1 P14902 2/20 0.36
TDO2 P48775 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL364862 0.89 EGFR (0.56) EGFRSRCKDM4EMAPTHPGD
SCHEMBL366454 0.83 EGFR (0.44) EGFRSRCKDM4EMAPTHPGD
SCHEMBL366300 0.82 CNR2 (0.38) EGFRSRCHPGDALDH1A1HDAC1
SCHEMBL366186 0.81 ALDH1A1 (0.39) EGFRSRCHPGDALDH1A1HSD17B10
SCHEMBL366536 0.80 EGFR (0.53) EGFRSRCKDM4EMAPTHPGD
SCHEMBL365488 0.80 PARP1 (0.41) EGFRSRCHPGDALDH1A1HDAC1
Potassium Ion SCHEMBL364977 0.78 EGFR (0.51) EGFRSRCKDM4EMAPTHPGD
SCHEMBL361357 0.78 EGFR (0.51) EGFRSRCKDM4EMAPTHPGD
SCHEMBL366838 0.78 ALDH1A1 (0.41) EGFRSRCKDM4EHPGDALDH1A1
SCHEMBL366239 0.78 PLA2G2A (0.41) HPGDALDH1A1ATMMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007007-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007007-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed