SCHEMBL3664825

SCHEMBL3664825

Nc1nccc(-c2ccc(N)c(OCCN3CCOCC3)c2)n1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 4/20 0.57
BCHE P06276 1/20 0.52
MAOA P21397 1/20 0.52
ACHE P22303 1/20 0.52
MAOB P27338 1/20 0.52
HSP90AA1 P07900 1/20 0.49
HSP90AB1 P08238 1/20 0.49
JAK2 O60674 2/20 0.48
MAPK13 O15264 1/20 0.48
MAPK12 P53778 1/20 0.48
MAPK11 Q15759 1/20 0.48
MAPK14 Q16539 1/20 0.48
KIT P10721 1/20 0.44
PIK3CA P42336 1/20 0.44
PDPK1 O15530 1/20 0.44
ADCY10 Q96PN6 1/20 0.44
TSHR P16473 1/20 0.44
HDAC1 Q13547 2/20 0.42
MET P08581 1/20 0.42
CCNA2 P20248 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3664819 0.86 KMO (0.59) KMOBCHEMAOAACHEMAOB
SCHEMBL4705549 0.77 ALDH1A1 (0.52) BCHEMAOAACHEMAOBJAK2
SCHEMBL3946646 0.76 CYP2D6 (0.50) BCHEMAOAACHEMAOBHSP90AA1
SCHEMBL15741737 0.74 ALDH1A1 (0.59) MAOBTSHR
SCHEMBL214175 0.74 KDM4E (0.53) MAOBMAPK14TSHR
SCHEMBL3656028 0.74 ROCK2 (0.60) KMOHSP90AA1PDPK1CCNA2CDK2
SCHEMBL1924882 0.73 LGMN (0.52) MAOBJAK2TSHR
Hydrochloric Acid SCHEMBL14784484 0.73 TSHR (0.51) MAOBTSHR
SCHEMBL4080135 0.72 LTA4H (0.56) BCHEMAOAACHEMAOB
SCHEMBL31125110 0.72 HRH2 (0.53) BCHEMAOAACHEMAOBTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2234618-A1 BENZOPYRANS AND ANALOGS AS RHO KINASE INHIBITORS The Scripps Research Institute (US) 2010-10-06 EP disclosed
WO-2009079008-A1 BENZOPYRANS AND ANALOGS AS RHO KINASE INHIBITORS FENG YANGBO (US) 2009-06-25 WO disclosed